SCHEMBL5407055

SCHEMBL5407055

Cc1cccc(CN(C)C(=O)c2ccccc2-c2ccccc2C(=O)N(CCCc2ccccc2)CCC(=O)O)n1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LTB4R2 Q9NPC1 2/20 0.41
LPAR1 Q92633 6/20 0.40
TDP1 Q9NUW8 1/20 0.39
POLB P06746 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TACR1 P25103 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5398682 0.95 KMT2A (0.44) KMT2AMEN1ALDH1A1LTB4R2TDP1
SCHEMBL5401005 0.91 KMT2A (0.48) KMT2AMEN1ALDH1A1LTB4R2LPAR1
SCHEMBL5412315 0.91 KMT2A (0.39) KMT2AMEN1ALDH1A1LPAR1TDP1
SCHEMBL5401118 0.90 KMT2A (0.39) KMT2AMEN1ALDH1A1TDP1POLB
SCHEMBL5392139 0.87 LPAR1 (0.41) KMT2AMEN1LPAR1TDP1SMN1; SMN2
SCHEMBL5401457 0.87 HTR2C (0.43) KMT2AMEN1ALDH1A1TDP1
SCHEMBL5405895 0.87 HCRTR1 (0.39) KMT2AMEN1ALDH1A1TDP1TACR1
SCHEMBL5404012 0.87 KDM4E (0.43) ALDH1A1TDP1POLBCYP2D6
SCHEMBL5404140 0.86 CA12 (0.46)
SCHEMBL5403805 0.86 RAB9A (0.44) KMT2AMEN1ALDH1A1LTB4R2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7285680-B2 β-alanine derivatives and the use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2007-10-23 US disclosed
US-20050256160-A1 Beta-alanine derivatives and the use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2005-11-17 US disclosed
EP-1533294-A1 BETA-ALANINE DERIVATIVE AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2005-05-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050256160-A1 Beta-alanine derivatives and the use thereof TGFB1, PML, APOB KMT2A 2451/4885MEN1 891/4885ALDH1A1 1256/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.