SCHEMBL540938

SCHEMBL540938

Nc1nc(Nc2ccccc2)nc(N(Cc2ccnc(F)c2)c2ccc(F)cc2)n1

nearest known ligand 0.91

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 13/20 0.91
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
HTT P42858 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MAPK1 P28482 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
HRH4 Q9H3N8 1/20 0.37
CDK9 P50750 1/20 0.37
GAA P10253 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1281689 0.95 KCNH3 (1.00) KCNH3NPC1RAB9ASMN1; SMN2MAPK1
SCHEMBL1923896 0.90 KCNH3 (0.81) KCNH3NPC1RAB9AHTTSMN1; SMN2
Hydrochloric Acid SCHEMBL540609 0.89 KCNH3 (0.82) KCNH3SMN1; SMN2CDK9
Hydrochloric Acid SCHEMBL540872 0.89 KCNH3 (0.82) KCNH3NPC1RAB9AHTTSMN1; SMN2
SCHEMBL1924291 0.88 KCNH3 (0.84) KCNH3NPC1RAB9AHTTMAPK1
Hydrochloric Acid SCHEMBL540943 0.87 KCNH3 (0.73) KCNH3NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL5017701 0.77 KCNH3 (0.62) KCNH3NPC1RAB9AHTTSMN1; SMN2
SCHEMBL1281719 0.72 KCNH3 (0.97) KCNH3
Hydrochloric Acid SCHEMBL541197 0.72 KCNH3 (1.00) KCNH3
SCHEMBL1923802 0.69 KCNH3 (0.88) KCNH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2413940-A1 COMPOSITIONS COMPRISING 2, 4, 6-TRIAMINO-1, 3, 5-TRIAZINE DERIVATIVES FOR TREATMENT OF SCHIZOPHRENIA Astellas Pharma Inc. (JP) 2012-02-08 EP disclosed
WO-2010114163-A1 COMPOSITIONS COMPRISING 2, 4, 6-TRIAMINO-1, 3, 5-TRIAZINE DERIVATIVES FOR TREATMENT OF SCHIZOPHRENIA ASTELLAS PHARMA INC. (JP) 2010-10-07 WO disclosed