SCHEMBL5409824

SCHEMBL5409824

Cc1c(Cl)cccc1S(=O)(=O)Nc1nnc(C(C)C)s1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 8/20 0.51
ALDH1A1 P00352 2/20 0.51
HSD17B10 Q99714 1/20 0.51
EDNRB P24530 2/20 0.49
EDNRA P25101 2/20 0.49
SLC40A1 Q9NP59 1/20 0.46
HSD17B1 P14061 2/20 0.45
HSD17B2 P37059 2/20 0.45
CCR4 P51679 1/20 0.44
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
GAA P10253 1/20 0.41
TSHR P16473 1/20 0.41
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5831160 0.87 HSD11B1 (0.46) HSD11B1ALDH1A1HSD17B10EDNRBEDNRA
SCHEMBL5399624 0.87 HSD11B1 (0.47) HSD11B1ALDH1A1HSD17B10EDNRBEDNRA
SCHEMBL5399619 0.87 HSD11B1 (0.47) HSD11B1ALDH1A1HSD17B10EDNRBEDNRA
SCHEMBL5389806 0.83 ALDH1A1 (0.47) HSD11B1ALDH1A1HSD17B10EDNRBEDNRA
SCHEMBL5389813 0.83 ALDH1A1 (0.47) HSD11B1ALDH1A1HSD17B10EDNRBEDNRA
SCHEMBL7059009 0.83 HSD11B1 (0.47) HSD11B1ALDH1A1HSD17B10EDNRBEDNRA
SCHEMBL5832114 0.82 HSD11B1 (0.48) HSD11B1ALDH1A1HSD17B10EDNRBEDNRA
SCHEMBL6624383 0.82 HSD11B1 (0.55) HSD11B1ALDH1A1HSD17B10EDNRBEDNRA
SCHEMBL5390611 0.81 MEN1 (0.64) HSD11B1ALDH1A1HSD17B10EDNRBEDNRA
SCHEMBL5410537 0.81 ALDH1A1 (0.44) HSD11B1ALDH1A1HSD17B10EDNRBEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070066614-A1 Ihibitors of 11-beta-hydroxy steroid dehydrogenase type 1 BIOVITRUM AB 2007-03-22 US claimed
US-7173030-B2 Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1 BIOVITRUM AB (SE) 2007-02-06 US claimed
EP-1631558-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE I BIOVITRUM AB (SE) 2006-03-08 EP claimed
US-20050009821-A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 BIOVITRUM AB 2005-01-13 US claimed
WO-2004103980-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE I BIOVITRUM AB (SE) 2004-12-02 WO claimed
US-20070066614-A1 Ihibitors of 11-beta-hydroxy steroid dehydrogenase type 1 BIOVITRUM AB 2007-03-22 US disclosed
US-7173030-B2 Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1 BIOVITRUM AB (SE) 2007-02-06 US disclosed
EP-1631558-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE I BIOVITRUM AB (SE) 2006-03-08 EP disclosed
US-20050009821-A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 BIOVITRUM AB 2005-01-13 US disclosed
WO-2004103980-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE I BIOVITRUM AB (SE) 2004-12-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050009821-A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 HSD11B1, HSD17B1, HSD11B2 HSD11B1 1/4885ALDH1A1 53/4885HSD17B10 22/4885
US-20070066614-A1 Ihibitors of 11-beta-hydroxy steroid dehydrogenase type 1 HSD11B1, HSD17B1, HSD17B11 HSD11B1 1/4885ALDH1A1 36/4885HSD17B10 16/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.