SCHEMBL5414397

SCHEMBL5414397

CO[C@]([C]=O)(c1ccccc1)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.38
TSHR P16473 2/20 0.38
CES1 P23141 1/20 0.38
KCNN4 O15554 1/20 0.37
PTPN1 P18031 1/20 0.35
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
MAPK1 P28482 2/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA5A P35218 1/20 0.34
CA9 Q16790 1/20 0.34
ALOX15 P16050 1/20 0.32
RORC P51449 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
KDM4E B2RXH2 2/20 0.32
GAA P10253 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL465653 1.00 ALDH1A1 (0.38) ALDH1A1TSHRCES1KCNN4PTPN1
SCHEMBL5161276 1.00 ALDH1A1 (0.38) ALDH1A1TSHRCES1KCNN4PTPN1
SCHEMBL13785277 0.81 ALDH1A1 (0.38) ALDH1A1TSHRCES1KCNN4PTPN1
SCHEMBL13785278 0.81 ALDH1A1 (0.38) ALDH1A1TSHRCES1KCNN4PTPN1
SCHEMBL7356506 0.80 ALDH1A1 (0.39) ALDH1A1TSHRKCNN4PTPN1NR1H2
SCHEMBL1401085 0.79 ALDH1A1 (0.35) ALDH1A1TSHRKCNN4PTPN1NR1H2
SCHEMBL4080546 0.76 KCNN4 (0.44) ALDH1A1TSHRCES1KCNN4PTPN1
SCHEMBL17091567 0.75 KCNN4 (0.34) ALDH1A1TSHRCES1KCNN4PTPN1
SCHEMBL7873896 0.71 ALDH1A1 (0.46) ALDH1A1TSHRCES1KCNN4MAPK1
SCHEMBL1229735 0.71 CES1 (0.42) ALDH1A1TSHRCES1KCNN4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0469887-B1 Acetamide derivatives ZENECA LTD (GB) 1994-12-14 EP claimed
US-5270342-A Acetamide derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-14 US claimed
EP-1663255-B1 WITHANAMIDE AND WITHANOLIDE COMPOSITIONS AND METHOD OF USE THEREOF UNIV MICHIGAN STATE (US) 2014-11-12 EP disclosed
US-7282593-B2 Withanamide and withanolide compositions and method of use thereof BOARD OF TRUSTEES OF MICHIGAN STATE UNIVERSITY (US) 2007-10-16 US disclosed
EP-1702910-A1 OCTAHYDRONAPHTHALENE DERIVATIVE AND MEDICINE Nippon Shinyaku Co., Ltd. (JP) 2006-09-20 EP disclosed
US-20050059727-A1 Withanamide and withanolide compositions and method of use thereof BOARD OF TRUSTEES OF MICHIGAN STATE UNIVERSITY (US) 2005-03-17 US disclosed
EP-0648130-B1 RADIOIODINATED BENZOVESAMICOL ANALOGS FOR CHOLINERGIC NERVE MAPPING UNIV MICHIGAN (US) 1998-12-30 EP disclosed
US-5430060-A Aldose reductase inhibitor ZENECA LIMITED (GB) 1995-07-04 US disclosed
US-5270342-A Acetamide derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-14 US disclosed
US-5077035-A Scintigraphic imaging of brain; Alzheimer*s diagnosis THE UNIVERSITY OF MICHIGAN (US) 1991-12-31 US disclosed
US-4772727-A Method of producing enantiomerically pure R-(+)-alpha-lipoic acid and S-(-)a DEGUSSA (DE) 1988-09-20 US disclosed
EP-0261336-A2 Process for the preparation of pure enantiomers of R-(+)-alpha-lipoic acid and S-(-)-alpha-lipoic acid (thioctic acid), and nonene or mesyl derivatives as intermediates therefor ASTA Medica Aktiengesellschaft (DE) 1988-03-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050059727-A1 Withanamide and withanolide compositions and method of use thereof ACHE, CYP51A1, HASPIN ALDH1A1 1849/4885TSHR 3754/4885CES1 344/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.