SCHEMBL5416163

SCHEMBL5416163

COCCNc1c(N)cnn1CCS(=O)(=O)O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
MAPT P10636 1/20 0.35
PTGER4 P35408 2/20 0.34
HTR4 Q13639 2/20 0.34
SYK P43405 3/20 0.33
KDM4E B2RXH2 1/20 0.33
HCAR3 P49019 1/20 0.33
CDK1 P06493 1/20 0.32
NCF1 P14598 1/20 0.32
LMNA P02545 2/20 0.31
PDE10A Q9Y233 1/20 0.31
JAK2 O60674 1/20 0.30
JAK3 P52333 1/20 0.30
CCNE2 O96020 1/20 0.30
CCNE1 P24864 1/20 0.30
CDK2 P24941 1/20 0.30
GSK3B P49841 1/20 0.30
MAPK8 P45983 1/20 0.30
MAPK9 P45984 1/20 0.30
MAPK10 P53779 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14445191 0.93 ALDH1A1 (0.34) ALDH1A1MAPTPTGER4HTR4SYK
SCHEMBL5423085 0.84 CDK1 (0.32) CDK1LMNA
SCHEMBL5413480 0.84 CDK1 (0.32) CDK1
SCHEMBL14445361 0.84 ALDH1A1 (0.38) ALDH1A1MAPTPTGER4KDM4EHCAR3
SCHEMBL5420777 0.83 CDK1 (0.33) CDK1
SCHEMBL14445366 0.81 ALDH1A1 (0.37) ALDH1A1MAPTPTGER4KDM4EHCAR3
SCHEMBL14445233 0.81 PTGER4 (0.38) ALDH1A1MAPTPTGER4KDM4EHCAR3
SCHEMBL5416172 0.80 CDK1 (0.32) CDK1
SCHEMBL14445194 0.78 CDK1 (0.32) CDK1
SCHEMBL14445304 0.78 ALDH1A1 (0.37) ALDH1A1MAPTPTGER4SYKKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7250063-B2 Diaminopyrazole derivatives and their use for oxidation dyeing of keratinous fibres L'OREAL (FR) 2007-07-31 US disclosed
US-7250063-B2 Diaminopyrazole derivatives and their use for oxidation dyeing of keratinous fibres L'OREAL (FR) 2007-07-31 US disclosed
US-7250063-B2 Diaminopyrazole derivatives and their use for oxidation dyeing of keratinous fibres L'OREAL (FR) 2007-07-31 US disclosed