SCHEMBL543248

SCHEMBL543248

O=C(Nc1ccc2[nH]nnc2c1)C1CC(=O)N(C2CCN(C(=O)O)CC2)C1

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL179133 0.88 PTPN2 (0.49) ALDH1A1SMN1; SMN2
SCHEMBL179131 0.88 ULK1 (0.50) ALDH1A1SMN1; SMN2KMT2A
SCHEMBL119244 0.84 P2RX7 (0.39) ALDH1A1SMN1; SMN2
SCHEMBL118397 0.84 ENPP2 (0.39) ALDH1A1SMN1; SMN2
SCHEMBL117356 0.84 ENPP2 (0.50)
SCHEMBL118794 0.83 ENPP2 (0.46)
SCHEMBL118895 0.82 HPGD (0.44) ALDH1A1SMN1; SMN2
SCHEMBL116941 0.82 MCHR1 (0.42) KMT2A
SCHEMBL16252470 0.82 ENPP2 (0.41) KMT2A
SCHEMBL118460 0.81 ENPP2 (0.42) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010115491-A2 PIPERIDINE AND PIPERAZINE DERIVATIVES AS AUTOTAXIN INHIBITORS MERCK PATENT GMBH (DE) 2010-10-14 WO claimed
EP-2414330-A2 PIPERIDINE AND PIPERAZINE DERIVATIVES AS AUTOTAXIN INHIBITORS Merck Patent GmbH (DE) 2012-02-08 EP disclosed
WO-2010115491-A2 PIPERIDINE AND PIPERAZINE DERIVATIVES AS AUTOTAXIN INHIBITORS MERCK PATENT GMBH (DE) 2010-10-14 WO disclosed