SCHEMBL543544

SCHEMBL543544

CC/C(=C\c1cccc2nn(C)cc12)C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.37
MTNR1B P49286 2/20 0.37
TBXAS1 P24557 2/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
GAA P10253 2/20 0.36
HTT P42858 2/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
CRHBP P24387 1/20 0.36
KMT2A Q03164 1/20 0.36
CRHR2 Q13324 1/20 0.36
USP2 O75604 1/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
ALOX15 P16050 1/20 0.34
ALOX12 P18054 1/20 0.34
HSD17B10 Q99714 1/20 0.34
USP7 Q93009 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL543545 1.00 MTNR1A (0.37) MTNR1AMTNR1BTBXAS1KDM4EALDH1A1
SCHEMBL543265 0.80 MAOA (0.33) MTNR1AMTNR1BTBXAS1LTB4RLTB4R2
SCHEMBL543225 0.80 MTNR1A (0.36) MTNR1AMTNR1BTBXAS1ALDH1A1MEN1
SCHEMBL543226 0.80 MTNR1A (0.36) MTNR1AMTNR1BTBXAS1ALDH1A1MEN1
SCHEMBL543266 0.80 MAOA (0.33) MTNR1AMTNR1BTBXAS1LTB4RLTB4R2
SCHEMBL544064 0.80 MTNR1A (0.36) MTNR1AMTNR1BTBXAS1EPHX2PPARG
SCHEMBL544065 0.80 MTNR1A (0.36) MTNR1AMTNR1BTBXAS1EPHX2PPARG
SCHEMBL2778053 0.75 NPC1 (0.45) KDM4EALDH1A1GAAHTTMEN1
SCHEMBL2778049 0.75 NPC1 (0.45) KDM4EALDH1A1GAAHTTMEN1
SCHEMBL543506 0.75 TBXAS1 (0.36) TBXAS1KDM4EALDH1A1GAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8110585-B2 Bicyclic compound and pharmaceutical use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-02-07 US disclosed