SCHEMBL5455762

SCHEMBL5455762

O=C1C2=C(CCCC2)C(=O)N1Cc1ccncc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1B1 Q16678 1/20 0.44
KDM4E B2RXH2 2/20 0.42
LMNA P02545 1/20 0.42
TNKS O95271 1/20 0.42
PARP1 P09874 1/20 0.42
PARP10 Q53GL7 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42
PARP2 Q9UGN5 1/20 0.42
PARP4 Q9UKK3 1/20 0.42
PARP3 Q9Y6F1 1/20 0.42
CA9 Q16790 3/20 0.40
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
FAAH O00519 1/20 0.39
MGLL Q99685 1/20 0.39
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 1/20 0.39
HPGD P15428 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2661082 0.80 KDM4E (0.57) CYP1B1KDM4ELMNAALDH1A1MEN1
SCHEMBL2662556 0.80 CASP3 (0.54) KDM4ELMNAALDH1A1MEN1HPGD
SCHEMBL6819071 0.78 MEN1 (0.46) CYP1B1CA9CA12CA1CA2
SCHEMBL41235 0.77 CA9 (0.53) CYP1B1CA9CA12CA1CA2
SCHEMBL24939710 0.76 PTGS1 (0.60) KDM4ELMNACA9CA1CA2
SCHEMBL5449610 0.76 CMA1 (0.64) KDM4EALDH1A1MEN1KMT2A
SCHEMBL6165776 0.74 CASP3 (0.62) CYP1B1KDM4ECA9CA12CA1
SCHEMBL8970292 0.74 ALDH1A1 (0.70) CYP1B1KDM4ELMNACA9CA12
SCHEMBL8970290 0.74 ALDH1A1 (0.70) CYP1B1KDM4ELMNACA9CA12
SCHEMBL14678510 0.71 MGLL (0.71) CYP1B1KDM4ECA9CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070117808-A1 Substituted Cycloalkylpyrrolones As Allosteric Modulators Of Glucokinase JANSSEN PHARMACEUTICA N.V. (BE) 2007-05-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070117808-A1 Substituted Cycloalkylpyrrolones As Allosteric Modulators Of Glucokinase GCKR, GCK, GALK1 CYP1B1 1325/4885KDM4E 1627/4885LMNA 4796/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.