SCHEMBL545967

SCHEMBL545967

CC(C)(C)N(CCc1cc(N)cc(C(F)(F)F)c1)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 14/20 0.43
MEN1 O00255 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
DHODH Q02127 1/20 0.33
NOS3 P29474 2/20 0.33
NOS1 P29475 2/20 0.33
NOS2 P35228 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL546112 0.86 TACR1 (0.41) TACR1MEN1HTTKMT2AL3MBTL1
SCHEMBL806193 0.76 NOS1 (0.49) TACR1NOS3NOS1NOS2
SCHEMBL1205533 0.76 MAOA (0.49) MEN1HTTKMT2AL3MBTL1
Hydrochloric Acid SCHEMBL787716 0.75 NOS1 (0.50) TACR1NOS3NOS1NOS2
SCHEMBL1845384 0.75 MEN1 (0.46) MEN1HTTKMT2AL3MBTL1
SCHEMBL5428175 0.74 TACR1 (0.52) TACR1
SCHEMBL27385426 0.74 TACR1 (0.42) TACR1MEN1KMT2A
SCHEMBL14257961 0.73 TACR1 (0.42) TACR1KMT2A
SCHEMBL28560207 0.72 EPHX1 (0.39) TACR1
SCHEMBL545287 0.72 NR1H2 (0.44) MEN1HTTKMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8110687-B2 Bicyclic compounds with kinase inhibitory activity MILLENNIUM PHARMACEUTICALS, INC. (US) 2012-02-07 US disclosed