SCHEMBL547802

SCHEMBL547802

CC1(C)COP(=O)(O)OC1c1ccccc1Cl

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.37
TP53 P04637 2/20 0.37
KMT2A Q03164 2/20 0.33
POLB P06746 1/20 0.33
TSHR P16473 1/20 0.33
RECQL P46063 1/20 0.33
KDM1A O60341 1/20 0.32
RCOR1 Q9UKL0 1/20 0.32
GAA P10253 2/20 0.32
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HTR2B P41595 1/20 0.31
CRHBP P24387 1/20 0.31
CRHR2 Q13324 1/20 0.31
ALDH1A1 P00352 2/20 0.31
OPRL1 P41146 1/20 0.30
KDM4E B2RXH2 1/20 0.30
GLA P06280 1/20 0.30
HPGD P15428 1/20 0.30
CASP1 P29466 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5678165 1.00 PTGS2 (0.37) PTGS2TP53KMT2APOLBTSHR
SCHEMBL29759482 1.00 PTGS2 (0.37) PTGS2TP53KMT2APOLBTSHR
SCHEMBL2026167 1.00 PTGS2 (0.37) PTGS2TP53KMT2APOLBTSHR
SCHEMBL29590612 1.00 PTGS2 (0.37) PTGS2TP53KMT2APOLBTSHR
SCHEMBL547467 0.89 HTR2A (0.35) TP53KMT2ATSHRGAAHTR2A
SCHEMBL1682788 0.86 TP53 (0.38) PTGS2TP53KMT2APOLBTSHR
SCHEMBL5678327 0.84 PTGS2 (0.35) PTGS2TP53KMT2APOLBTSHR
SCHEMBL28361354 0.84 HTR5A (0.31) HTR2AHTR2C
SCHEMBL28194083 0.84 HTR5A (0.31) HTR2AHTR2C
SCHEMBL28194084 0.84 HTR5A (0.31) HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 98 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107602464-B Method for preparing biaryl quinoline antibiotics by optical resolution 宜昌人福药业有限责任公司 2020-02-18 CN claimed
CN-104876856-A Method for preparing (R)-(+)-3-piperidinamine dihydrochloride by using resolution method HEBEI KAILIANG BIOTECHNOLOGY CO LTD 2015-09-02 CN claimed
CN-104829459-A Splitting method for preparing (R)-(+)-1-naphthyl ethylamine HEBEI CHIRAL CHEMISTRY AND BIOTECHNOLOGY CO LTD 2015-08-12 CN claimed
CN-103755582-B Preparation method according to D-serine through splitting method UNIV HEBEI SCIENCE & TECH 2015-04-08 CN claimed
CN-103755582-A Preparation method according to D-serine through splitting method UNIV HEBEI SCIENCE & TECH 2014-04-30 CN claimed
CN-102070469-B Resolution method for preparing optically pure metoprolol UNIV HEBEI SCIENCE & TECH 2013-11-20 CN claimed
CN-101792398-B Method for preparing optical pure p-hydroxy phenyl glycine by separation method UNIV HEBEI SCIENCE & TECH 2013-06-26 CN claimed
CN-102070469-A Resolution method for preparing optically pure metoprolol UNIV HEBEI SCIENCE & TECH 2011-05-25 CN claimed
CN-101792398-A Method for preparing optical pure p-hydroxy phenyl glycine by separation method HEBEI UNIVERSITY OF SCIENCE & TECHNOLOGY 2010-08-04 CN claimed
US-5663354-A Process for preparing enantiomerically pure 6-[(4-chlorophenyl) (1H-1,2,4-triazol-1-yl) methyl]-1-methyl-1H-benzotrizole JANSSEN PHARMACEUTICA, N.V. (BE) 1997-09-02 US claimed
EP-0668861-A1 PROCESS FOR PREPARING ENANTIOMERICALLY PURE 6- (4-CHLOROPHENYL)(1H --TRIAZOL-1,2,4-TRIAZOL-1-YL)METHYL]-1-METHYL-1H --BENZOTRIAZOLE JANSSEN PHARMACEUTICA N.V. (BE) 1995-08-30 EP claimed
WO-1994011364-A1 PROCESS FOR PREPARING ENANTIOMERICALLY PURE 6-[(4-CHLOROPHENYL)(1H^_-TRIAZOL-1,2,4-TRIAZOL-1-YL)METHYL]-1-METHYL-1H^_-BENZOTRIAZOLE JANSSEN PHARMACEUTICA N.V. (BE) 1994-05-26 WO claimed
CN-110317212-B Synthesis of polycyclic carbamoylpyridone compounds 吉利德科学公司 2022-10-21 CN disclosed
EP-4045615-A1 AN INDUSTRIAL PROCESS FOR RESOLUTION OF CHLOCYPHOS Hikal Limited (IN) 2022-08-24 EP disclosed
CN-114394983-A Synthesis of polycyclic carbamoylpyridone compounds 吉利德科学公司 2022-04-26 CN disclosed
WO-2021074778-A1 AN INDUSTRIAL PROCESS FOR RESOLUTION OF CHLOCYPHOS HIKAL LIMITED (IN) 2021-04-22 WO disclosed
US-4968837-A Resolution of racemic mixtures ETHYL CORPORATION (US) 1990-11-06 US disclosed
WO-1989012445-A1 METHOD AND COMPOSITIONS FOR TREATMENT OF PARKINSONISM SYNDROME IN MAMMALS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-12-28 WO disclosed
US-4885308-A ADMINISTERING DOPAMINERGIC TETRALIN DERIVATIVE NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-12-05 US disclosed
EP-0180276-B1 DIOXAPHOSPHORINANES, THEIR PREPARATION AND USE FOR RESOLVING OPTICALLY ACTIVE COMPOUNDS STAMICARBON B.V. (NL) 1988-12-28 EP disclosed