SCHEMBL4599464

SCHEMBL4599464

Fc1cccc(C(Cl)OCc2ccccc2)c1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.45
TDO2 P48775 1/20 0.45
CNR2 P34972 1/20 0.44
SLC6A9 P48067 1/20 0.44
SLC6A5 Q9Y345 1/20 0.44
AGXT P21549 2/20 0.42
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
PPARG P37231 1/20 0.39
PPARA Q07869 1/20 0.39
TACR1 P25103 1/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
SLC6A3 Q01959 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL547986 0.82 SLC6A2 (0.47) IDO1AGXTMEN1KMT2ATACR1
SCHEMBL28534097 0.81 CHRNB2 (0.45) IDO1AGXTMEN1KMT2ATACR1
SCHEMBL6205189 0.81 CNR2 (0.48) IDO1TDO2CNR2SLC6A9SLC6A5
SCHEMBL6205190 0.81 CNR2 (0.48) IDO1TDO2CNR2SLC6A9SLC6A5
SCHEMBL6035746 0.78 IDO1 (0.43) IDO1TDO2CNR2SLC6A9SLC6A5
SCHEMBL27502909 0.75 ALOX5 (0.50) KMT2APPARGPPARASLC6A2SLC6A4
SCHEMBL6181884 0.73 CHRNB2 (0.63) IDO1TDO2AGXTMEN1KMT2A
SCHEMBL22785928 0.72 CA1 (0.47) IDO1TDO2CNR2SLC6A9SLC6A5
SCHEMBL7817242 0.72 MAOB (0.54) KMT2A
SCHEMBL28528002 0.71 CHRNB2 (0.45) AGXTMEN1KMT2ATACR1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910363-A2 HIV INTEGRASE INHIBITORS SmithKline Beecham Corporation (US) 2008-04-16 EP disclosed
WO-2007019098-A2 HIV INTEGRASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2007-02-15 WO disclosed
EP-1720856-A2 HIV INTEGRASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2006-11-15 EP disclosed
WO-2005077050-A2 HIV INTEGRASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2005-08-25 WO disclosed