SCHEMBL5481197

SCHEMBL5481197

CCCc1c(I)cccc1C(N)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
NR1I2 O75469 1/20 0.40
CHRM2 P08172 1/20 0.40
CYP3A4 P08684 1/20 0.40
ADRA2A P08913 1/20 0.40
OPRK1 P41145 1/20 0.40
HTR2B P41595 1/20 0.40
SLC6A3 Q01959 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 3/20 0.39
HSD17B10 Q99714 3/20 0.39
HPGD P15428 2/20 0.39
HTT P42858 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
PDPK1 O15530 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2964481 0.87 PARP1 (0.45) PARP1LMNAMAPTMEN1KMT2A
SCHEMBL5685703 0.81 ALDH1A1 (0.42) PARP1LMNAMAPTMEN1KMT2A
SCHEMBL4235369 0.81 CXCR5 (0.49) PARP1LMNAMAPTMEN1KMT2A
SCHEMBL3352032 0.81 PARP1 (0.41) PARP1LMNAMAPTMEN1KMT2A
Charcoal, Activated SCHEMBL9341326 0.79 PARP1 (0.40) PARP1LMNAMAPTMEN1KMT2A
SCHEMBL5483010 0.79 PARP1 (0.40) PARP1LMNAMAPTMEN1KMT2A
SCHEMBL21439307 0.79 MAPK8 (0.44) PARP1LMNAMAPTMEN1KMT2A
SCHEMBL6314578 0.79 PARP1 (0.40) PARP1LMNAMAPTMEN1KMT2A
SCHEMBL28273750 0.79 ALDH1A1 (0.41) PARP1LMNAMAPTMEN1KMT2A
SCHEMBL144959 0.77 PARP1 (0.44) PARP1LMNAMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1763509-A1 ALPHA-HELICAL MIMETICS THE WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH (AU) 2007-03-21 EP disclosed
WO-2006002474-A1 ALPHA-HELICAL MIMETICS THE WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH (AU) 2006-01-12 WO disclosed