SCHEMBL5483010

SCHEMBL5483010

CCCc1c(Br)cccc1C(N)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 2/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
NR1I2 O75469 1/20 0.40
CHRM2 P08172 1/20 0.40
CYP3A4 P08684 1/20 0.40
ADRA2A P08913 1/20 0.40
OPRK1 P41145 1/20 0.40
HTR2B P41595 1/20 0.40
SLC6A3 Q01959 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
METAP2 P50579 1/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
HPGD P15428 2/20 0.39
HSD17B10 Q99714 2/20 0.39
HTT P42858 1/20 0.38
PARP2 Q9UGN5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28204079 0.90 LMNA (0.44) PARP1LMNAMAPTKMT2AMEN1
SCHEMBL2964481 0.87 PARP1 (0.45) PARP1LMNAMAPTKMT2AMEN1
SCHEMBL5701955 0.86 PARP1 (0.45) PARP1LMNAMAPTKMT2AMEN1
Hydrochloric Acid SCHEMBL27970367 0.84 PARP1 (0.44) PARP1LMNAMAPTKMT2AMEN1
SCHEMBL6469520 0.84 F2R (0.41) KMT2AMEN1ALDH1A1F2R
SCHEMBL2729495 0.84 PRNP (0.44) ALDH1A1KDM4EHPGDHSD17B10F2R
SCHEMBL3352032 0.81 PARP1 (0.41) PARP1LMNAMAPTKMT2AMEN1
SCHEMBL5685703 0.81 ALDH1A1 (0.42) PARP1LMNAMAPTKMT2AMEN1
SCHEMBL4235369 0.81 CXCR5 (0.49) PARP1LMNAMAPTKMT2AMEN1
SCHEMBL6637803 0.80 GAA (0.44) LMNAKMT2AMEN1SLC6A3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1763509-A1 ALPHA-HELICAL MIMETICS THE WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH (AU) 2007-03-21 EP disclosed
WO-2006002474-A1 ALPHA-HELICAL MIMETICS THE WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH (AU) 2006-01-12 WO disclosed