SCHEMBL5481366

SCHEMBL5481366

CS(=O)(=O)OCC1(CC#Cc2ccc(OC(F)(F)F)cc2)CCC1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.39
ACACB O00763 1/20 0.37
SLC6A4 P31645 7/20 0.36
SLC6A3 Q01959 6/20 0.36
SLC6A2 P23975 2/20 0.36
KIF11 P52732 1/20 0.36
PTGS1 P23219 1/20 0.34
HSD11B1 P28845 1/20 0.33
MMP14 P50281 2/20 0.32
PDE2A O00408 2/20 0.32
MMP1 P03956 1/20 0.32
MMP13 P45452 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
BCHE P06276 1/20 0.32
ACHE P22303 1/20 0.32
MMP2 P08253 1/20 0.32
MMP9 P14780 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5484802 0.81 ACACB (0.36) ACACBSLC6A4SLC6A3SLC6A2HSD11B1
SCHEMBL5482423 0.80 LMNA (0.41) ACACBSLC6A4SLC6A3SLC6A2
SCHEMBL3871947 0.75 ACACB (0.39) PTGS2ACACBSLC6A4SLC6A3KIF11
SCHEMBL28768495 0.74 ACACB (0.41) ACACBSLC6A4SLC6A3MMP2MMP9
SCHEMBL5484157 0.72 POLB (0.42) ACACBSLC6A4SLC6A3PDE2AMEN1
SCHEMBL5485919 0.70 PPARD (0.40)
SCHEMBL5481378 0.70 ACACB (0.38) PTGS2ACACBSLC6A4SLC6A3SLC6A2
SCHEMBL16841023 0.68 ACACB (0.44) ACACBSLC6A4SLC6A3SLC6A2MEN1
SCHEMBL7008210 0.68 KIF11 (0.46) PTGS2SLC6A4SLC6A3KIF11MMP14
SCHEMBL14671190 0.67 KDM4E (0.39) MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7253192-B2 Phenyl derivatives comprising an acetylene group HOFFMANN-LA ROCHE INC. (US) 2007-08-07 US disclosed
US-20060004091-A1 Phenyl derivatives comprising an acetylene group F. HOFFMANN-LA ROCHE AG (CH) 2006-01-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060004091-A1 Phenyl derivatives comprising an acetylene group PPARD, PPARA, PPARG PTGS2 718/4885ACACB 47/4885SLC6A4 4267/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.