SCHEMBL5483719

SCHEMBL5483719

Cc1c(N2CCN(C(=O)O)CC2=O)nnn1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.47
TP53 P04637 3/20 0.41
ALOX12 P18054 1/20 0.41
ALDH1A1 P00352 3/20 0.39
PFKFB3 Q16875 3/20 0.38
LMNA P02545 2/20 0.37
KDM4E B2RXH2 2/20 0.37
GAA P10253 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PDK2 Q15119 1/20 0.36
P2RX7 Q99572 2/20 0.35
SCD5 Q86SK9 1/20 0.35
PTGS2 P35354 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ALPI P09923 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14582539 0.89 HTT (0.43) HTTTP53ALOX12ALDH1A1LMNA
SCHEMBL2887702 0.86 CSNK1E (0.45) HTTTP53ALOX12GAAPDK2
SCHEMBL2893886 0.86 GPR119 (0.42) HTTTP53ALOX12ALDH1A1LMNA
SCHEMBL2894092 0.85 MEN1 (0.45) HTTALDH1A1LMNAKDM4EGAA
SCHEMBL2891520 0.85 P2RX7 (0.46) P2RX7
SCHEMBL2890817 0.81 HTT (0.52) HTTTP53ALOX12ALDH1A1LMNA
SCHEMBL5481400 0.80 P2RX7 (0.37) P2RX7
SCHEMBL15988360 0.77 KMT2A (0.52) ALDH1A1P2RX7SCD5KMT2A
SCHEMBL2893237 0.75 HTT (0.43) HTTTP53ALOX12ALDH1A1LMNA
SCHEMBL14582401 0.73 HTT (0.50) HTTTP53ALOX12ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1764362-A1 BIARYL DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 2007-03-21 EP disclosed