Metyrapone

Metyrapone

SCHEMBL5484012

CC(C)(C(=O)c1cccnc1)c1cccnc1.Cl.Cl

nearest known ligand 0.97

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

CYP11B1

The experimentally established mechanism targets of Metyrapone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 known ✓ P15538 1/20 0.97
TDP1 Q9NUW8 2/20 0.97
LMNA P02545 1/20 0.97
CYP1A2 P05177 1/20 0.97
CYP3A4 P08684 1/20 0.97
CYP11B2 P19099 1/20 0.97
ALDH1A1 P00352 3/20 0.50
APP P05067 1/20 0.50
GAA P10253 1/20 0.50
HCAR3 P49019 1/20 0.50
HCAR2 Q8TDS4 1/20 0.50
THRB P10828 1/20 0.49
F7 P08709 1/20 0.49
F3 P13726 1/20 0.49
SARM1 Q6SZW1 1/20 0.49
SIRT2 Q8IXJ6 1/20 0.49
SIRT6 Q8N6T7 1/20 0.49
SIRT1 Q96EB6 1/20 0.49
SIRT3 Q9NTG7 1/20 0.49
SIRT5 Q9NXA8 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Metyrapone SCHEMBL29462551 0.98 TDP1 (1.00) TDP1LMNACYP1A2CYP3A4CYP11B1
Metyrapone SCHEMBL637432 0.98 TDP1 (1.00) TDP1LMNACYP1A2CYP3A4CYP11B1
Metyrapone SCHEMBL29917903 0.98 TDP1 (1.00) TDP1LMNACYP1A2CYP3A4CYP11B1
SCHEMBL12260655 0.90 CYP3A4 (0.84) TDP1LMNACYP1A2CYP3A4CYP11B1
Metyrapone SCHEMBL30807826 0.88 LMNA (0.81) TDP1LMNACYP1A2CYP3A4CYP11B1
Metyrapone SCHEMBL667561 0.88 LMNA (0.81) TDP1LMNACYP1A2CYP3A4CYP11B1
Metyrapone SCHEMBL667560 0.88 LMNA (0.81) TDP1LMNACYP1A2CYP3A4CYP11B1
Metyrapone SCHEMBL7020159 0.85 LMNA (0.74) TDP1LMNACYP1A2CYP3A4CYP11B1
SCHEMBL31703901 0.80 LMNA (0.69) TDP1LMNACYP1A2CYP3A4CYP11B1
SCHEMBL800635 0.80 LMNA (0.69) TDP1LMNACYP1A2CYP3A4CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007062198-A1 METHODS TO ACCELERATE THE ISOLATION OF NOVEL CELL STRAINS FROM PLURIPOTENT STEM CELLS AND CELLS OBTAINED THEREBY ADVANCED CELL TECHNOLOGY, INC. (US) 2007-05-31 WO disclosed