SCHEMBL5486378

SCHEMBL5486378

O=C1OCCN1c1cc(Cl)cc(N2CCOC2=O)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKAG1 P54619 1/20 0.40
PRKAA1 Q13131 1/20 0.40
PRKAB1 Q9Y478 1/20 0.40
IDH1 O75874 2/20 0.40
TNKS O95271 1/20 0.37
F10 P00742 1/20 0.36
CMA1 P23946 1/20 0.36
MAP2K1 Q02750 1/20 0.36
EGLN2 Q96KS0 1/20 0.35
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
NAAA Q02083 2/20 0.35
KDM1A O60341 2/20 0.35
MAOA P21397 2/20 0.35
MAOB P27338 2/20 0.35
RCOR1 Q9UKL0 2/20 0.35
DGAT1 O75907 2/20 0.34
KDM1B Q8NB78 1/20 0.34
CCNC P24863 1/20 0.34
CDK8 P49336 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11595049 0.96 IDH1 (0.40) PRKAG1PRKAA1PRKAB1IDH1TNKS
SCHEMBL5174949 0.82 PIK3CA (0.38) IDH1TNKSMAP2K1EGLN2DGAT1
SCHEMBL13167913 0.82 HSD11B1 (0.47) TNKSF10CMA1NAAAKDM1A
SCHEMBL13167926 0.78 HSP90AA1 (0.39) IDH1TNKSEGLN2DGAT1CCNC
SCHEMBL5800891 0.78 PIK3CA (0.43) IDH1TNKSEGLN2CCNCCDK8
SCHEMBL21723494 0.78 SLC6A2 (0.48) CMA1ADRB1ALDH1A1
SCHEMBL30980936 0.78 DRD2 (0.40) IDH1F10CMA1DRD2DRD3
SCHEMBL15499081 0.75 PKM (0.48) CMA1CCNCCDK8ALDH1A1HSD17B10
SCHEMBL8349969 0.74 BPTF (0.43) TNKSCMA1EGLN2DGAT1CCNC
SCHEMBL26298453 0.74 EGLN2 (0.40) IDH1TNKSCMA1MAP2K1EGLN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1787684-B1 New couplers HENKEL AG & CO KGAA (DE) 2016-01-20 EP claimed
EP-1787684-A2 New couplers Henkel Kommanditgesellschaft auf Aktien (DE) 2007-05-23 EP claimed
EP-1787684-B1 New couplers HENKEL AG & CO KGAA (DE) 2016-01-20 EP disclosed
EP-1787684-A2 New couplers Henkel Kommanditgesellschaft auf Aktien (DE) 2007-05-23 EP disclosed
EP-1787684-A2 New couplers Henkel Kommanditgesellschaft auf Aktien (DE) 2007-05-23 EP disclosed