SCHEMBL5486737

SCHEMBL5486737

OC[C@H](O)c1cccc(Br)c1F

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 3/20 0.41
ADRA2B P18089 3/20 0.41
ADRA2C P18825 3/20 0.41
ADRB1 P08588 1/20 0.41
ADRB3 P13945 1/20 0.41
ADRA1A P35348 2/20 0.34
ADRB2 P07550 1/20 0.34
ADRA1B P35368 1/20 0.34
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
GABRA1 P14867 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
SLC18A3 Q16572 1/20 0.31
SIGMAR1 Q99720 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2947197 1.00 ADRA2A (0.41) ADRA2AADRA2BADRA2CADRB1ADRB3
SCHEMBL22051464 0.79 CES2 (0.35) ADRA2AADRA2BADRA2CADRB1ADRB3
SCHEMBL31376555 0.79 SLC18A3 (0.43) SLC18A3SIGMAR1
SCHEMBL29811265 0.79 SLC18A3 (0.43) SLC18A3SIGMAR1
SCHEMBL4975851 0.79 SLC18A3 (0.43) SLC18A3SIGMAR1
SCHEMBL16959073 0.79 GABRA1 (0.31) ADRA2AADRA2BADRA2CADRB1ADRB3
SCHEMBL611730 0.79 ADRA2A (0.37) ADRA2AADRA2BADRA2CADRB1ADRB3
SCHEMBL14837162 0.79 ADRA2A (0.37) ADRA2AADRA2BADRA2CADRB1ADRB3
SCHEMBL30910218 0.76 CES2 (0.33) ADRA2AADRA2BADRA2CADRB1ADRB3
SCHEMBL30967943 0.76 HTR2C (0.37) ADRA2AADRA2BADRA2CADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1752452-A9 PROPANE-1,3-DIONE DERIVATIVE OR ITS SALT Astellas Pharma Inc. (JP) 2007-12-12 EP disclosed
EP-1752452-A1 PROPANE-1,3-DIONE DERIVATIVE OR ITS SALT Astellas Pharma Inc. (JP) 2007-02-14 EP disclosed