SCHEMBL5487018

SCHEMBL5487018

CCOC(=O)c1ccc2cc(-c3cccnc3)ccc2c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 6/20 0.74
CYP19A1 P11511 5/20 0.74
CYP11B1 P15538 5/20 0.74
MMP2 P08253 1/20 0.64
MMP13 P45452 1/20 0.64
MMP14 P50281 1/20 0.64
CYP17A1 P05093 3/20 0.53
SLC2A1 P11166 1/20 0.53
ACHE P22303 1/20 0.52
KDM4E B2RXH2 3/20 0.51
ALDH1A1 P00352 3/20 0.51
MAPT P10636 3/20 0.51
NPSR1 Q6W5P4 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
MKNK1 Q9BUB5 2/20 0.50
MKNK2 Q9HBH9 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5735824 0.86 MKNK1 (0.59) CYP11B2CYP19A1CYP11B1MMP2MMP13
SCHEMBL4509922 0.85 CYP11B2 (1.00) CYP11B2CYP19A1CYP11B1CYP17A1SLC2A1
SCHEMBL1895643 0.81 CYP2C9 (0.57) MMP2MMP13MMP14SLC2A1KDM4E
SCHEMBL13712389 0.81 CYP11B2 (0.72) CYP11B2CYP19A1CYP11B1CYP17A1SLC2A1
SCHEMBL6041578 0.81 CA12 (0.51) CYP11B2CYP19A1CYP11B1KDM4EALDH1A1
SCHEMBL29613178 0.81 CA12 (0.51) CYP11B2CYP19A1CYP11B1KDM4EALDH1A1
SCHEMBL23484192 0.81 CA12 (0.56) CYP11B2CYP19A1CYP11B1MMP2MMP13
SCHEMBL10028690 0.80 ALDH1A1 (0.56) MMP2MMP13MMP14SLC2A1KDM4E
SCHEMBL4027305 0.79 MMP2 (0.60) CYP11B2CYP19A1CYP11B1MMP2MMP13
SCHEMBL707407 0.78 CA12 (0.67) SLC2A1KDM4EALDH1A1MAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1853261-A1 SELECTIVE INHIBITORS OF HUMAN CORTICOSTEROID SYNTHASES Universität des Saarlandes (DE) 2007-11-14 EP disclosed
WO-2006092430-A1 SELECTIVE INHIBITORS OF HUMAN CORTICOSTEROID SYNTHASES Universität des Saarlandes (DE) 2006-09-08 WO disclosed