SCHEMBL5487498

SCHEMBL5487498

COc1cc(-n2nnc(NS(N)(=O)=O)c2-c2cccc3[nH]c(C(C)C)nc23)c(O)cc1O

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.33
MGAM O43451 1/20 0.32
GAA P10253 1/20 0.32
SI P14410 1/20 0.32
MGAM2 Q2M2H8 1/20 0.32
HTR3A P46098 7/20 0.31
HTR4 Q13639 7/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1148514 0.81 HCRTR1 (0.37) GAA
SCHEMBL1342905 0.80 CCNB2 (0.36) GAA
SCHEMBL1344647 0.73 NR1I2 (0.32)
SCHEMBL1344644 0.72 KIF11 (0.39)
SCHEMBL2596697 0.72 MGAM (0.34) PARP1MGAMGAASIMGAM2
SCHEMBL1148440 0.69 ALDH1A1 (0.37) GAA
SCHEMBL1148557 0.67 PDE4D (0.37)
SCHEMBL1148837 0.66 ALDH1A1 (0.36)
SCHEMBL1344291 0.65 NR1I2 (0.41) GAA
SCHEMBL1148817 0.63 ALDH1A1 (0.39) L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817295-A1 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY Synta Pharmaceuticals Corporation (US) 2007-08-15 EP claimed
WO-2006055760-A9 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY SYNTA PHARMACEUTICALS CORP (US) 2006-09-21 WO claimed
WO-2006055760-A1 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY SYNTA PHARMACEUTICALS CORP. (US) 2006-05-26 WO claimed