SCHEMBL2596697

SCHEMBL2596697

COc1cc(-c2nnc(OS(N)(=O)=O)n2-c2cccc3[nH]c(C(C)C)nc23)c(O)cc1O

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MGAM O43451 3/20 0.34
GAA P10253 3/20 0.34
SI P14410 3/20 0.34
MGAM2 Q2M2H8 3/20 0.34
PARP1 P09874 5/20 0.34
CDK2 P24941 3/20 0.33
PRKCZ Q05513 3/20 0.33
HTR3A P46098 3/20 0.32
HTR4 Q13639 3/20 0.32
KCNN4 O15554 1/20 0.31
DHODH Q02127 1/20 0.31
HSP90AA1 P07900 1/20 0.30
HSP90AB1 P08238 1/20 0.30
CDK4 P11802 1/20 0.30
CCNA2 P20248 1/20 0.30
CCND1 P24385 1/20 0.30
CCND3 P30281 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL930673 0.79 SLC37A4 (0.37) GAAKCNN4HSP90AA1HSP90AB1
SCHEMBL421146 0.79 CCNB2 (0.34)
SCHEMBL15472986 0.76 APLNR (0.32) KCNN4HSP90AA1HSP90AB1
SCHEMBL931915 0.74 TUBB4A (0.38) GAAHSP90AA1HSP90AB1
SCHEMBL5487498 0.72 PARP1 (0.33) MGAMGAASIMGAM2PARP1
SCHEMBL15468253 0.68 HSP90AA1 (0.40) GAAKCNN4HSP90AA1HSP90AB1
SCHEMBL16604230 0.67 TUBB4A (0.38) HSP90AA1HSP90AB1
SCHEMBL930691 0.66 MEN1 (0.36) GAAKCNN4HSP90AA1HSP90AB1
SCHEMBL445050 0.65 APLNR (0.37)
SCHEMBL1305403 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011146801-A1 FORMULATION AND DOSING OF HSP90 INHIBITORY COMPOUNDS SYNTA PHARMACEUTICALS CORP. (US) 2011-11-24 WO claimed
WO-2011146801-A1 FORMULATION AND DOSING OF HSP90 INHIBITORY COMPOUNDS SYNTA PHARMACEUTICALS CORP. (US) 2011-11-24 WO disclosed