SCHEMBL54882

SCHEMBL54882

Cn1c2ccc(S(=O)(=O)Cl)cc2c(=O)c2cc(S(=O)(=O)Cl)ccc21

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIK3CG P48736 2/20 0.47
PARG Q86W56 5/20 0.41
PKM P14618 2/20 0.40
HTT P42858 2/20 0.40
MITF O75030 1/20 0.40
LMNA P02545 1/20 0.40
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
ATM Q13315 1/20 0.39
TAS2R14 Q9NYV8 3/20 0.39
HCRTR1 O43613 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
TP53 P04637 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29558921 1.00 PIK3CG (0.47) PIK3CGPARGPKMHTTMITF
SCHEMBL3761642 0.92 ATM (0.51) PIK3CGHTTNPC1RAB9AMEN1
SCHEMBL17715367 0.87 PIK3CG (0.39) PIK3CGPARGPKMHTTMITF
SCHEMBL27651563 0.83 MAPT (0.54) PIK3CGHTTMEN1KMT2AATM
SCHEMBL20855010 0.82 PIK3CG (0.47) PIK3CGPARGPKMHTTMITF
SCHEMBL17832062 0.81 PIK3CG (0.72) PIK3CGPARGPKMHTTMITF
SCHEMBL26090948 0.80 PARG (0.64) PIK3CGPARGPKMHTTMITF
SCHEMBL17825124 0.79 PARG (0.61) PIK3CGPARGPKMHTTMITF
SCHEMBL5865904 0.77 PARG (0.47) PIK3CGPARGTP53
SCHEMBL1278983 0.76 KDM4E (0.58) PKMHTTLMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230159762-A1 NIR TO SWIR FLUORESCENT COMPOUNDS FOR IMAGING AND DETECTION REVVITY HEALTH SCIENCES, INC. 2023-05-25 US disclosed
US-20230159762-A1 NIR TO SWIR FLUORESCENT COMPOUNDS FOR IMAGING AND DETECTION REVVITY HEALTH SCIENCES, INC. 2023-05-25 US disclosed
US-11549017-B2 NIR to SWIR fluorescent compounds for imaging and detection PERKINELMER HEALTH SCIENCES, INC. (US) 2023-01-10 US disclosed
CN-108314663-B Derivatives of fluorene, anthracene, xanthene, dibenzosuberone and acridine and uses thereof 多格伍德药品公司 2022-05-13 CN disclosed
WO-2019067180-A1 NIR TO SWIR FLUORESCENT COMPOUNDS FOR IMAGING AND DETECTION PERKINELMER HEALTH SCIENCES, INC. (US) 2019-04-04 WO disclosed
US-20190100654-A1 NIR TO SWIR FLUORESCENT COMPOUNDS FOR IMAGING AND DETECTION REVVITY HEALTH SCIENCES, INC. 2019-04-04 US disclosed
US-9446021-B2 Derivatives of fluorene, anthracene, xanthene, dibenzosuberone and acridine and uses thereof DOGWOOD PHARMACEUTICALS, INC. (US) 2016-09-20 US disclosed
US-9446021-B2 Derivatives of fluorene, anthracene, xanthene, dibenzosuberone and acridine and uses thereof DOGWOOD PHARMACEUTICALS, INC. (US) 2016-09-20 US disclosed
US-9446021-B2 Derivatives of fluorene, anthracene, xanthene, dibenzosuberone and acridine and uses thereof DOGWOOD PHARMACEUTICALS, INC. (US) 2016-09-20 US disclosed
EP-2152258-B1 DERIVATIVES OF FLUORENE, ANTHRACENE, XANTHENE, DIBENZOSUBERONE AND ACRIDINE AND USES THEREOF AVALON PHARMACEUTICALS (US) 2016-05-04 EP disclosed
US-8129519-B2 Derivatives of fluorene, anthracene, xanthene, dibenzosuberone and acridine and uses thereof ALLERGAN SALES, LLC 2012-03-06 US disclosed
US-8129519-B2 Derivatives of fluorene, anthracene, xanthene, dibenzosuberone and acridine and uses thereof ALLERGAN SALES, LLC 2012-03-06 US disclosed
WO-2010082912-A1 DERIVATIVES OF MULTI-RING AROMATIC COMPOUNDS AND USES AS ANTI-TUMOR AGENTS AVALON PHARMACEUTICALS (US) 2010-07-22 WO disclosed
WO-2010082912-A1 DERIVATIVES OF MULTI-RING AROMATIC COMPOUNDS AND USES AS ANTI-TUMOR AGENTS AVALON PHARMACEUTICALS (US) 2010-07-22 WO disclosed
US-20100137354-A1 DERIVATIVES OF FLUORENE, ANTHRACENE, XANTHENE, DIBENZOSUBERONE AND ACRIDINE AND USES THEREOF ALLERGAN SALES, LLC 2010-06-03 US disclosed
US-20100137354-A1 DERIVATIVES OF FLUORENE, ANTHRACENE, XANTHENE, DIBENZOSUBERONE AND ACRIDINE AND USES THEREOF ALLERGAN SALES, LLC 2010-06-03 US disclosed
US-20100137354-A1 DERIVATIVES OF FLUORENE, ANTHRACENE, XANTHENE, DIBENZOSUBERONE AND ACRIDINE AND USES THEREOF ALLERGAN SALES, LLC 2010-06-03 US disclosed
EP-2152258-A1 DERIVATIVES OF FLUORENE, ANTHRACENE, XANTHENE, DIBENZOSUBERONE AND ACRIDINE AND USES THEREOF Avalon Pharmaceuticals (US) 2010-02-17 EP disclosed
WO-2008140792-A1 DERIVATIVES OF FLUORENE, ANTHRACENE, XANTHENE, DIBENZOSUBERONE AND ACRIDINE AND USES THEREOF AVALON PHARMACEUTICALS (US) 2008-11-20 WO disclosed
WO-2008140792-A1 DERIVATIVES OF FLUORENE, ANTHRACENE, XANTHENE, DIBENZOSUBERONE AND ACRIDINE AND USES THEREOF AVALON PHARMACEUTICALS (US) 2008-11-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100137354-A1 DERIVATIVES OF FLUORENE, ANTHRACENE, XANTHENE, DIBENZOSUBERONE AND ACRIDINE AND USES THEREOF WNT1, CTNND1, CTNNB1 PIK3CG 3284/4885PARG 4086/4885PKM 4502/4885
US-11549017-B2 NIR to SWIR fluorescent compounds for imaging and detection SMARCD1, SMARCE1, SMARCB1 PIK3CG 2889/4885PARG 1087/4885PKM 2856/4885
US-20190100654-A1 NIR TO SWIR FLUORESCENT COMPOUNDS FOR IMAGING AND DETECTION SMARCD1, SMARCE1, SMARCB1 PIK3CG 2889/4885PARG 1087/4885PKM 2856/4885
US-20230159762-A1 NIR TO SWIR FLUORESCENT COMPOUNDS FOR IMAGING AND DETECTION SMARCD1, SMARCE1, SMARCB1 PIK3CG 2889/4885PARG 1087/4885PKM 2856/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.