SCHEMBL5488302

SCHEMBL5488302

CC(C)c1ccc(N)cn1.CC(C)c1ccc([N+](=O)[O-])cn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.47
MAPT P10636 7/20 0.43
KMT2A Q03164 4/20 0.43
MEN1 O00255 3/20 0.43
RAB9A P51151 2/20 0.43
NPC1 O15118 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ADRA2A P08913 2/20 0.42
ADRA2B P18089 2/20 0.42
ADRA2C P18825 2/20 0.42
SLC2A1 P11166 1/20 0.42
LMNA P02545 3/20 0.41
CYP1A2 P05177 1/20 0.41
GAA P10253 1/20 0.41
CHRNA7 P36544 1/20 0.40
HSP90AA1 P07900 1/20 0.39
CXCR5 P32302 1/20 0.39
APLNR P35414 1/20 0.39
CCR6 P51684 1/20 0.39
GFER P55789 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL397421 0.90 MAPT (0.49) ALDH1A1MAPTKMT2AMEN1RAB9A
Formamide SCHEMBL28333185 0.86 SLC2A1 (0.46) ALDH1A1MAPTKMT2AMEN1RAB9A
SCHEMBL5371 0.81 CHRNA7 (0.44) ALDH1A1MAPTKMT2AMEN1RAB9A
Ammonia Solution, Strong SCHEMBL7429890 0.79 ADRA2A (0.45) ALDH1A1MAPTKMT2AMEN1RAB9A
SCHEMBL28062195 0.77 GAA (0.45) ALDH1A1MAPTKMT2AMEN1RAB9A
SCHEMBL19089741 0.77 CYP1A2 (0.49) ALDH1A1MAPTKMT2AMEN1RAB9A
SCHEMBL4434207 0.76 ALDH1A1 (0.52) ALDH1A1MAPTKMT2AMEN1RAB9A
SCHEMBL8466648 0.76 ALDH1A1 (0.52) ALDH1A1MAPTKMT2AMEN1ADRA2A
SCHEMBL18078274 0.74 MAPT (0.54) ALDH1A1MAPTKMT2AMEN1RAB9A
SCHEMBL3973866 0.73 ADRA2A (0.46) ALDH1A1MAPTKMT2AMEN1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773816-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2007-04-18 EP disclosed
WO-2006002421-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-01-05 WO disclosed