SCHEMBL5488534

SCHEMBL5488534

Nc1ncc(-c2ccc(C(=O)N3CCCC3CN3CCCC3)cc2)nc1OCc1c(Cl)cccc1Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 3/20 1.00
MET P08581 13/20 0.73
ATR Q13535 1/20 0.60
ALK Q9UM73 2/20 0.53
HRH3 Q9Y5N1 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30453716 1.00 CSF1R (1.00) CSF1RMETATRALKHRH3
SCHEMBL487740 1.00 CSF1R (1.00) CSF1RMETATRALKHRH3
SCHEMBL30453712 0.88 CSF1R (0.79) CSF1RMETATRALKHRH3
SCHEMBL488002 0.88 CSF1R (0.79) CSF1RMETATRALKHRH3
SCHEMBL30452641 0.86 CSF1R (0.75) CSF1RMETATRALKHRH3
SCHEMBL488141 0.86 CSF1R (0.75) CSF1RMETATRALKHRH3
SCHEMBL488668 0.86 CSF1R (0.75) CSF1RMETATRALKHRH3
SCHEMBL30453070 0.86 CSF1R (0.75) CSF1RMETATRALKHRH3
SCHEMBL488143 0.86 CSF1R (0.75) CSF1RMETATRALKHRH3
SCHEMBL5488939 0.85 CSF1R (0.75) CSF1RMETATRALKHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7230098-B2 2-amino- pyridines and pyrazines additionally substituted witn one or more carbocyclic or heterocyclic groups, e.g., 4-[6-amino-5-(2,6-dichloro-benzyloxy)-pyridin-3-yl]-phenol, for treating many kinds of cancer SUGEN, INC. (US) 2007-06-12 US disclosed
US-20050009840-A1 2-amino- pyridines and pyrazines additionally substituted witn one or more carbocyclic or heterocyclic groups, e.g., 4-[6-amino-5-(2,6-dichloro-benzyloxy)-pyridin-3-yl]-phenol, for treating many kinds of cancer SUGEN, INC. 2005-01-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050009840-A1 2-amino- pyridines and pyrazines additionally substituted witn one or more carbocyclic or heterocyclic groups, e.g., 4-[6-amino-5-(2,6-dichloro-benzyloxy)-pyridin-3-yl]-phenol, for treating many kinds of cancer MET, ERBB2, CDK4 CSF1R 1027/4885MET 1/4885ATR 1572/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.