SCHEMBL5488544

SCHEMBL5488544

NC(=O)C1(C(=O)O)C=Cc2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.36
THRB P10828 1/20 0.36
TSHR P16473 2/20 0.34
LMNA P02545 1/20 0.34
MAPK1 P28482 1/20 0.34
SCN4A P35499 1/20 0.34
SCN5A Q14524 1/20 0.34
SCN9A Q15858 1/20 0.34
KIF11 P52732 5/20 0.34
POLB P06746 1/20 0.33
CYP3A4 P08684 1/20 0.33
PARP1 P09874 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C19 P33261 1/20 0.33
RECQL P46063 1/20 0.33
BLM P54132 1/20 0.33
PMP22 Q01453 1/20 0.33
HSD17B10 Q99714 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HSD11B1 P28845 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6055589 0.89 THRB (0.41) TDP1THRBKIF11HSD11B1AKR1C1
SCHEMBL27970747 0.74 THRB (0.38) TDP1THRBTSHRLMNAMAPK1
SCHEMBL31325165 0.74 THRB (0.38) TDP1THRBTSHRLMNAMAPK1
SCHEMBL31181875 0.73 CCKAR (0.38) TSHRLMNAMAPK1SCN4ASCN5A
SCHEMBL29118949 0.72 ALDH1A1 (0.33) TDP1POLBMAPTBLMHSD17B10
SCHEMBL28032107 0.72 THRB (0.44) TDP1THRBKIF11HSD11B1AKR1C1
SCHEMBL14232376 0.70 CCKAR (0.39) TDP1THRBKIF11HSD11B1AKR1C1
SCHEMBL28807690 0.70 KMT2A (0.34) TDP1THRBPOLBMAPTHSD17B10
SCHEMBL30990090 0.69 KDM4E (0.37) TDP1THRBMAPTHSD11B1
SCHEMBL7031865 0.68 KMT2A (0.35) TDP1THRBTSHRLMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007516982-A 2007-06-28 JP claimed
EP-1694410-A2 CYCLOPROPANE COMPOUNDS AND PHARMACEUTICAL USE THEREOF Japan Tobacco, Inc. (JP) 2006-08-30 EP claimed
WO-2005058884-A2 CYCLOPROPANE COMPOUNDS AND PHARMACEUTICAL USE THEREOF JAPAN TOBACCO INC. (JP) 2005-06-30 WO claimed
EP-1694410-A2 CYCLOPROPANE COMPOUNDS AND PHARMACEUTICAL USE THEREOF Japan Tobacco, Inc. (JP) 2006-08-30 EP disclosed
WO-2005058884-A2 CYCLOPROPANE COMPOUNDS AND PHARMACEUTICAL USE THEREOF JAPAN TOBACCO INC. (JP) 2005-06-30 WO disclosed