SCHEMBL5490989

SCHEMBL5490989

CS(=O)(=O)c1ccc([C@@H](CC=O)c2cc(F)cc(Cl)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.46
PTGS2 P35354 13/20 0.42
EPAS1 Q99814 2/20 0.40
EPHX2 P34913 3/20 0.39
ESR2 Q92731 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5494676 1.00 CCR5 (0.46) CCR5PTGS2EPAS1EPHX2ESR2
SCHEMBL4915625 0.91 EPHX2 (0.43) CCR5PTGS2EPHX2ESR2
SCHEMBL4915630 0.91 EPHX2 (0.43) CCR5PTGS2EPHX2ESR2
SCHEMBL27643617 0.82 AKR1C3 (0.44) CCR5PTGS2EPHX2
SCHEMBL5459229 0.82 AKR1C3 (0.44) CCR5PTGS2EPHX2
SCHEMBL20902116 0.79 MDM2 (0.39)
SCHEMBL4977528 0.77 PTGS2 (0.44) PTGS2ESR2
SCHEMBL4975056 0.77 PTGS2 (0.44) PTGS2ESR2
SCHEMBL4904275 0.77 EPHX2 (0.52) CCR5PTGS2EPHX2ESR2
SCHEMBL4904265 0.77 EPHX2 (0.52) CCR5PTGS2EPHX2ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7294636-B2 Chemical compounds ASTRAZENECA AB (SE) 2007-11-13 US disclosed
CN-1784393-A Chemical compounds ASTRAZENECA AB (SE) 2006-06-07 CN disclosed