SCHEMBL5491963

SCHEMBL5491963

CCc1ccc(N)cc1N.CCc1ccc(N)cc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 2/20 0.50
MAPT P10636 6/20 0.45
ALDH1A1 P00352 6/20 0.45
GAA P10253 5/20 0.45
KDM4E B2RXH2 4/20 0.45
POLB P06746 3/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
HTT P42858 2/20 0.45
USP2 O75604 2/20 0.45
TP53 P04637 1/20 0.45
CASP7 P55210 1/20 0.45
ATM Q13315 1/20 0.45
TSHR P16473 2/20 0.45
MAPK1 P28482 1/20 0.45
PRKCI P41743 1/20 0.42
TDP1 Q9NUW8 4/20 0.41
ACHE P22303 1/20 0.41
GFER P55789 1/20 0.39
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL396816 1.00 CASP1 (0.50) CASP1MAPTALDH1A1GAAKDM4E
SCHEMBL29414153 1.00 CASP1 (0.50) CASP1MAPTALDH1A1GAAKDM4E
SCHEMBL395438 0.84 PRKCI (0.47) CASP1MAPTALDH1A1GAAKDM4E
SCHEMBL29738343 0.84 PRKCI (0.47) CASP1MAPTALDH1A1GAAKDM4E
SCHEMBL398586 0.83 GAA (0.46) CASP1MAPTALDH1A1GAAKDM4E
SCHEMBL94119 0.82 ALDH1A1 (0.50) CASP1MAPTALDH1A1GAAKDM4E
SCHEMBL27770925 0.82 CASP1 (0.42) CASP1MAPTALDH1A1GAAKDM4E
SCHEMBL30227490 0.82 ALDH1A1 (0.50) CASP1MAPTALDH1A1GAAKDM4E
Hydrochloric Acid SCHEMBL8667386 0.81 GAA (0.48) CASP1MAPTALDH1A1GAAKDM4E
SCHEMBL10890416 0.81 CASP1 (0.46) CASP1MAPTALDH1A1GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773816-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2007-04-18 EP disclosed
WO-2006002421-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-01-05 WO disclosed