SCHEMBL5494098

SCHEMBL5494098

CON(C(=O)c1cc(NC(=O)c2cc(F)cc(N3CCCC3)c2)cnc1C)c1ccc(NCC2CC2)nc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 4/20 0.42
MAPK14 Q16539 7/20 0.39
SMO Q99835 1/20 0.39
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
MAPT P10636 2/20 0.35
TSHR P16473 2/20 0.35
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
OPRK1 P41145 1/20 0.34
ITGB3 P05106 1/20 0.34
ITGB1 P05556 1/20 0.34
ITGAV P06756 1/20 0.34
ITGA5 P08648 1/20 0.34
ITGB5 P18084 1/20 0.34
MAPK13 O15264 1/20 0.34
MAPK12 P53778 1/20 0.34
MAPK11 Q15759 1/20 0.34
LCK P06239 1/20 0.34
KDR P35968 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5490030 0.99 CRHR1 (0.42) CRHR1MAPK14SMONPC1RAB9A
SCHEMBL4551483 0.95 MAPK14 (0.39) CRHR1MAPK14SMOMAPK13MAPK12
SCHEMBL4551537 0.95 MAPK14 (0.39) CRHR1MAPK14SMOMAPK13MAPK12
SCHEMBL14534448 0.91 HCAR3 (0.40) MAPK14SMONPC1RAB9AMAPT
SCHEMBL4551763 0.90 MAPK14 (0.39) MAPK14SMONPC1RAB9AMAPT
SCHEMBL5494096 0.89 CRHR1 (0.42) CRHR1ITGB3ITGB1ITGAVITGA5
SCHEMBL5495529 0.89 MAPK14 (0.39) MAPK14SMONPC1RAB9AMAPT
SCHEMBL5490026 0.89 CRHR1 (0.42) CRHR1ITGB3ITGB1ITGAVITGA5
SCHEMBL5490107 0.87 MAPK14 (0.39) MAPK14SMONPC1RAB9AMAPT
SCHEMBL5490598 0.87 CRHR1 (0.50) CRHR1MAPK14SMONPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007056016-A2 BISAMIDE CYTOKINE INHIBITORS KEMIA, INC. (US) 2007-05-18 WO disclosed
WO-2007056016-A2 BISAMIDE CYTOKINE INHIBITORS KEMIA, INC. (US) 2007-05-18 WO disclosed