SCHEMBL5494699

SCHEMBL5494699

COc1ccc(N(c2ccc(C=Cc3cccc(C)c3)cc2)c2ccc(OC)cc2)cc1.COc1cccc(N(c2ccc(C=Cc3ccccc3)cc2)c2cccc(OC)c2)c1

nearest known ligand 0.68

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RELA Q04206 5/20 0.68
TRPA1 O75762 1/20 0.53
NFE2L2 Q16236 2/20 0.48
APP P05067 1/20 0.48
CYP19A1 P11511 1/20 0.48
CYP1A1 P04798 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP1B1 Q16678 2/20 0.46
NQO2 P16083 1/20 0.45
MAPT P10636 1/20 0.44
THRB P10828 1/20 0.44
ACHE P22303 1/20 0.44
CHRNA7 P36544 1/20 0.44
SNCA P37840 1/20 0.44
TRPM8 Q7Z2W7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5494696 1.00 RELA (0.68) RELATRPA1NFE2L2APPCYP19A1
SCHEMBL5494942 0.91 RELA (0.82) RELATRPA1NFE2L2APPCYP19A1
SCHEMBL5494946 0.91 RELA (0.82) RELATRPA1NFE2L2APPCYP19A1
SCHEMBL10015726 0.90 RELA (0.69) RELANFE2L2APPCYP19A1CYP1A1
SCHEMBL16167740 0.90 RELA (0.69) RELANFE2L2APPCYP19A1CYP1A1
SCHEMBL16311931 0.90 RELA (0.69) RELANFE2L2APPCYP19A1CYP1A1
SCHEMBL5491678 0.89 RELA (0.58) RELATRPA1NFE2L2CYP19A1CYP1A1
SCHEMBL5491677 0.89 RELA (0.58) RELATRPA1NFE2L2CYP19A1CYP1A1
SCHEMBL8943695 0.88 RELA (0.56) RELATRPA1NFE2L2CYP19A1CYP1A1
SCHEMBL8943692 0.88 RELA (0.56) RELATRPA1NFE2L2CYP19A1CYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7276627-B2 One pot sequential reactions and novel products produced thereby IOWA STATE UNIVERSITY RESEARCH FOUNDATION, INC. (US) 2007-10-02 US disclosed
US-20060224017-A1 One pot sequential reactions and novel products produced thereby IOWA STATE UNIVERSITY RESEARCH FOUNDATION, INC. 2006-10-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060224017-A1 One pot sequential reactions and novel products produced thereby PNMT, CYP1A1, TERT RELA 1503/4885TRPA1 1677/4885NFE2L2 446/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.