SCHEMBL5497823

SCHEMBL5497823

CC(C)(C)OC(=O)NCCC(=O)NCCc1cn[nH]c1NC(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.43
IDO1 P14902 5/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
NQO2 P16083 1/20 0.39
CYP3A4 P08684 1/20 0.39
NPSR1 Q6W5P4 1/20 0.37
BCHE P06276 1/20 0.37
ALDH1A1 P00352 1/20 0.36
GFER P55789 1/20 0.36
CKS1B P61024 1/20 0.36
SKP1 P63208 1/20 0.36
SKP2 Q13309 1/20 0.36
KDM4E B2RXH2 3/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6557087 0.88 SIGMAR1 (0.42) SIGMAR1IDO1NQO2CYP3A4NPSR1
SCHEMBL6557081 0.87 NPSR1 (0.43) SIGMAR1IDO1CYP3A4NPSR1BCHE
SCHEMBL6385864 0.84 BCHE (0.40) SIGMAR1IDO1NQO2CYP3A4NPSR1
SCHEMBL6387372 0.79 CKS1B (0.42) SIGMAR1IDO1CA1CA2CYP3A4
SCHEMBL6559029 0.76 SIGMAR1 (0.37) SIGMAR1IDO1BCHECKS1BSKP1
SCHEMBL5497821 0.75 SIGMAR1 (0.38) SIGMAR1IDO1CA1CA2CYP3A4
SCHEMBL25048413 0.74 CA1 (0.60) SIGMAR1IDO1CA1CA2KDM4E
SCHEMBL6385861 0.71 BCHE (0.40) SIGMAR1IDO1NQO2NPSR1BCHE
SCHEMBL31505697 0.69 MALT1 (0.51) SIGMAR1IDO1CA1CA2NQO2
SCHEMBL5497926 0.69 TLR7 (0.38) SIGMAR1IDO1CA1CA2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1556389-B1 CEPHEM COMPOUNDS ASTELLAS PHARMA INC (JP) 2007-07-25 EP disclosed