SCHEMBL5498128

SCHEMBL5498128

COc1cccc(CC2(O)CCNCC2)c1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.49
CYP2D6 P10635 2/20 0.45
USP2 O75604 1/20 0.45
POLB P06746 1/20 0.42
BRD4 O60885 1/20 0.41
CYP1A2 P05177 1/20 0.40
CHRM2 P08172 1/20 0.40
SLC6A4 P31645 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 2/20 0.39
TP53 P04637 1/20 0.39
APOBEC3A P31941 1/20 0.39
CTDSP1 Q9GZU7 1/20 0.39
APOBEC3G Q9HC16 1/20 0.39
DRD2 P14416 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20070372 0.87 SIGMAR1 (0.56) SIGMAR1CYP2D6USP2POLBCYP1A2
Hydrochloric Acid SCHEMBL20138396 0.85 SIGMAR1 (0.55) SIGMAR1CYP2D6USP2SLC6A4ALDH1A1
SCHEMBL25596166 0.73 SIGMAR1 (0.41) SIGMAR1CYP2D6USP2CYP1A2SLC6A4
SCHEMBL27932886 0.73 GAA (0.51) SIGMAR1CYP2D6USP2CYP1A2CHRM2
SCHEMBL16657601 0.73 FPR2 (0.53) SIGMAR1CYP2D6USP2SLC6A4DRD2
Hydrochloric Acid SCHEMBL28086905 0.72 FPR2 (0.52) SIGMAR1CYP2D6USP2SLC6A4APOBEC3A
SCHEMBL7290612 0.72 LMNA (0.46) SIGMAR1SLC6A4MEN1KMT2A
SCHEMBL7446267 0.71 POLB (0.56) POLBBRD4KDM4EALDH1A1TP53
Hydrochloric Acid SCHEMBL20137513 0.71 LMNA (0.49) SIGMAR1SLC6A4MEN1KMT2A
SCHEMBL8401996 0.71 CYP1A2 (0.76) CYP2D6USP2POLBCYP1A2CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1768958-A1 NEW DISUBSTITUTED PHENYLPIPERIDINES AS MODULATORS OF DOPAMINE AND SEROTONIN NEUROTRANSMISSION A. CARLSSON RESEARCH AB (SE) 2007-04-04 EP disclosed
WO-2005121088-A1 NEW DISUBSTITUTED PHENYLPIPERIDINES AS MODULATORS OF DOPAMINE AND SEROTONIN NEUROTRANSMISSION A. CARLSSON RESEARCH AB (SE) 2005-12-22 WO disclosed