SCHEMBL5499152

SCHEMBL5499152

CCC(C)OP(=O)(O)C(F)(F)c1ccc(C(CC(=O)NCCCCc2ccccc2)NS(=O)(=O)c2ccccc2)cc1Br

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
HPGD P15428 1/20 0.40
KMT2A Q03164 1/20 0.40
BDKRB1 P46663 1/20 0.36
MMP2 P08253 3/20 0.36
MMP7 P09237 3/20 0.36
MMP9 P14780 3/20 0.36
MMP13 P45452 3/20 0.36
MMP1 P03956 2/20 0.36
MMP3 P08254 2/20 0.36
GAA P10253 1/20 0.35
THRB P10828 1/20 0.34
MAPK1 P28482 1/20 0.34
FAAH O00519 1/20 0.34
TACR1 P25103 1/20 0.34
NLRP3 Q96P20 1/20 0.34
MMP8 P22894 1/20 0.34
MMP14 P50281 1/20 0.34
ATM Q13315 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3743225 0.80 CNR1 (0.37) ALDH1A1MMP2MMP7MMP9MMP13
SCHEMBL3738015 0.80 MLYCD (0.48) ALDH1A1HPGDNLRP3L3MBTL1MAPT
SCHEMBL3737791 0.78 TRPV1 (0.44) HPGD
SCHEMBL3738515 0.77 TRPV1 (0.47) ALDH1A1HPGDKMT2A
SCHEMBL3737636 0.76 CA1 (0.42) ALDH1A1HPGDKMT2AMAPTCA1
SCHEMBL3736646 0.75 LMNA (0.41) ALDH1A1HPGDKMT2AL3MBTL1MAPT
SCHEMBL7594249 0.74 PTPN1 (0.36) ALDH1A1ATML3MBTL1
SCHEMBL3746413 0.74 ALDH1A1 (0.44) ALDH1A1MMP2MMP7MMP9MMP13
SCHEMBL3743393 0.73 ALDH1A1 (0.47) ALDH1A1HPGDKMT2AGAAMAPT
SCHEMBL7598030 0.73 PTPN1 (0.37) ALDH1A1ATML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1812012-A2 PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF Ceptyr, Inc. (US) 2007-08-01 EP disclosed
WO-2006055525-A2 PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF CEPTYR, INC. (US) 2006-05-26 WO disclosed