SCHEMBL5500516

SCHEMBL5500516

CN(C)CCCOc1ccc(-c2ccc(CC3CCCC(N4CCCC4=O)C3)c(Cl)c2)cc1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ATM Q13315 4/20 0.41
ESR1 P03372 1/20 0.39
ATR Q13535 1/20 0.38
HRH3 Q9Y5N1 5/20 0.36
LSS P48449 1/20 0.36
UTS2R Q9UKP6 4/20 0.36
PIK3CA P42336 1/20 0.35
SLC6A4 P31645 2/20 0.34
PARP1 P09874 1/20 0.34
CXCR1 P25024 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5499707 0.99 ATM (0.40) ATMESR1ATRHRH3LSS
SCHEMBL5503492 0.96 ESR1 (0.43) ATMESR1ATRHRH3LSS
Hydrochloric Acid SCHEMBL5500694 0.95 ESR1 (0.42) ATMESR1ATRHRH3LSS
SCHEMBL5503554 0.91 PARP1 (0.34) ATMESR1ATRHRH3UTS2R
SCHEMBL5500808 0.86 ESR1 (0.37) ESR1HRH3PIK3CAPARP1
SCHEMBL5500801 0.82 CHEK2 (0.37)
SCHEMBL5504232 0.82 CTSS (0.36)
Hydrochloric Acid SCHEMBL5500756 0.82 CHEK2 (0.36)
SCHEMBL5499827 0.81 P2RX7 (0.34)
SCHEMBL5506180 0.80 AAK1 (0.34) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1807072-A1 CYCLOALKYL LACTAM DERIVATIVES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE 1 ELI LILLY AND COMPANY (US) 2007-07-18 EP claimed
WO-2006049952-A1 CYCLOALKYL LACTAM DERIVATIVES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE 1 ELI LILLY AND COMPANY (US) 2006-05-11 WO claimed