SCHEMBL5500808

SCHEMBL5500808

Cc1cc(OCCN(C)C)ccc1-c1ccc(CC2CCCC(N3CCCC3=O)C2)c(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.37
PIK3CA P42336 1/20 0.37
PRKDC P78527 1/20 0.37
MMP2 P08253 1/20 0.34
MMP3 P08254 1/20 0.34
PARP1 P09874 2/20 0.34
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
FFAR1 O14842 1/20 0.33
SCN9A Q15858 1/20 0.32
TNKS O95271 1/20 0.32
BTK Q06187 1/20 0.31
KMT2A Q03164 2/20 0.31
PRMT5 O14744 1/20 0.31
WDR77 Q9BQA1 1/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5503554 0.96 PARP1 (0.34) ESR1PIK3CAPRKDCPARP1FFAR1
SCHEMBL5503492 0.90 ESR1 (0.43) ESR1PIK3CAPRKDCPARP1KDM4E
Hydrochloric Acid SCHEMBL5500694 0.90 ESR1 (0.42) ESR1PIK3CAPRKDCPARP1KDM4E
SCHEMBL5503919 0.88 HTR1A (0.37) FFAR1SCN9AHRH3
SCHEMBL5500516 0.86 ATM (0.41) ESR1PIK3CAPARP1HRH3
Hydrochloric Acid SCHEMBL5499707 0.86 ATM (0.40) ESR1PIK3CAPARP1HRH3
Hydrochloric Acid SCHEMBL5500185 0.85 SSTR2 (0.36)
SCHEMBL5499853 0.83 SCN9A (0.37) ESR1SCN9A
SCHEMBL3544979 0.79 PIK3CA (0.38) ESR1PIK3CAPRKDCMMP2MMP3
SCHEMBL5501522 0.77 CYP11B2 (0.36) SCN9ABTKPRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1807072-A1 CYCLOALKYL LACTAM DERIVATIVES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE 1 ELI LILLY AND COMPANY (US) 2007-07-18 EP claimed
WO-2006049952-A1 CYCLOALKYL LACTAM DERIVATIVES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE 1 ELI LILLY AND COMPANY (US) 2006-05-11 WO claimed