SCHEMBL5500828

SCHEMBL5500828

NC(=O)NCCc1ccc(O)c(O)c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.70
HSD17B10 Q99714 4/20 0.70
KDM4E B2RXH2 4/20 0.70
HIF1A Q16665 3/20 0.70
ALDH1A1 P00352 3/20 0.70
LMNA P02545 3/20 0.70
BLM P54132 3/20 0.70
HPGD P15428 2/20 0.70
PTGS1 P23219 2/20 0.70
CA1 P00915 2/20 0.58
CA2 P00918 2/20 0.58
CA9 Q16790 2/20 0.58
CA7 P43166 1/20 0.58
CA14 Q9ULX7 1/20 0.58
ALOX15 P16050 3/20 0.58
MAPK1 P28482 3/20 0.58
TP53 P04637 2/20 0.58
THPO P40225 2/20 0.58
CYP1A2 P05177 1/20 0.58
TSHR P16473 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7361910 0.86 MAPT (0.66) MAPTHSD17B10KDM4EHIF1AALDH1A1
SCHEMBL109163 0.85 MAPT (0.74) MAPTHSD17B10KDM4EHIF1AALDH1A1
SCHEMBL7105545 0.85 MAPT (0.74) MAPTHSD17B10KDM4EHIF1AALDH1A1
SCHEMBL6420228 0.84 MAPT (0.72) MAPTHSD17B10KDM4EHIF1AALDH1A1
SCHEMBL30252290 0.83 MAPT (0.66) MAPTHSD17B10KDM4EHIF1AALDH1A1
SCHEMBL28976197 0.83 MAPT (0.66) MAPTHSD17B10KDM4EHIF1AALDH1A1
SCHEMBL29782210 0.82 MAPT (0.64) MAPTHSD17B10KDM4EHIF1AALDH1A1
SCHEMBL25380895 0.82 MAPT (0.70) MAPTHSD17B10KDM4EHIF1AALDH1A1
SCHEMBL109158 0.82 MAPT (0.73) MAPTHSD17B10KDM4EHIF1AALDH1A1
SCHEMBL328568 0.82 MAPT (1.00) MAPTHSD17B10KDM4EHIF1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1751097-A1 SUBSTITUTED N-ARYL BENZAMIDES AND RELATED COMPOUNDS FOR TREATMENT OF AMYLOID DISEASES AND SYNUCLEINOPATHIES Proteotech, Inc. (US) 2007-02-14 EP claimed
WO-2005113489-A1 SUBSTITUTED N-ARYL BENZAMIDES AND RELATED COMPOUNDS FOR TREATMENT OF AMYLOID DISEASES AND SYNUCLEINOPATHIES PROTEOTECH, INC. (US) 2005-12-01 WO claimed
US-20230355843-A1 INJECTABLE CUSHIONING HYDROGELS SUPRA B B.V. (NL) 2023-11-09 US disclosed
US-20230012485-A1 ADHESIVE DEVICE FOR BIOMEDICAL APPLICATIONS AND METHODS OF USE THEREOF SUNNYBROOK HEALTH SCIENCES CENTRE (CA) 2023-01-19 US disclosed
US-20230001046-A1 BIOCOMPATIBLE ADHESIVES AND METHODS OF MANUFACTURE THEREOF GOVERNING COUNCIL UNIV TORONTO (CA) 2023-01-05 US disclosed