SCHEMBL5501166

SCHEMBL5501166

CC1OCCc2c(O)cccc21

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 3/20 0.41
DRD2 P14416 4/20 0.40
HTR1A P08908 3/20 0.40
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15319916 0.80 ADRA2A (0.39) DRD1
SCHEMBL3715028 0.79 GID4 (0.41) DRD1DRD2
SCHEMBL1660824 0.72 DRD2 (0.50) DRD2HTR1AESR1ESR2
SCHEMBL19661160 0.72 DRD2 (0.50) DRD2HTR1AESR1ESR2
SCHEMBL1598610 0.70 DRD2 (0.45) DRD1DRD2ESR1ESR2
SCHEMBL23921624 0.69 HTR2A (0.43)
SCHEMBL660714 0.69 HTR2A (0.43)
SCHEMBL15384214 0.69 DRD2 (0.48) DRD2HTR1AESR1ESR2
SCHEMBL1660087 0.69 ADRA2A (0.50) DRD2HTR1AESR1ESR2
SCHEMBL15576799 0.69 KCNJ1 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1749001-A1 3-PIPERIDINYLISOCHROMAN-5-OLS AS DOPAMINE AGONISTS Aventis Pharmaceuticals, Inc. (US) 2007-02-07 EP disclosed
WO-2005111025-A1 3-PIPERIDINYLISOCHROMAN-5-OLS AS DOPAMINE AGONISTS AVENTIS PHARMACEUTICALS INC. (US) 2005-11-24 WO disclosed