SCHEMBL5504141

SCHEMBL5504141

C#C[C@H]1O[C@@H](n2cnc3c(NC4CCC(F)C4)ncnc32)[C@@H]2OC(C)(C)O[C@@H]21

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PI4KA P42356 1/20 0.41
PI4K2B Q8TCG2 1/20 0.41
PI4K2A Q9BTU6 1/20 0.41
PI4KB Q9UBF8 1/20 0.41
ADORA3 P0DMS8 5/20 0.41
ADORA1 P30542 5/20 0.41
ADORA2A P29274 3/20 0.41
ADORA2B P29275 2/20 0.41
PMP22 Q01453 1/20 0.40
GAA P10253 1/20 0.40
HTT P42858 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
SLC29A1 Q99808 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5504146 1.00 PI4KA (0.41) PI4KAPI4K2BPI4K2API4KBADORA3
SCHEMBL5507495 0.90 ADORA3 (0.41) PI4KAPI4K2BPI4K2API4KBADORA3
SCHEMBL5507489 0.90 ADORA3 (0.41) PI4KAPI4K2BPI4K2API4KBADORA3
SCHEMBL5509240 0.88 TSHR (0.52) ADORA3ADORA1ADORA2AADORA2BPMP22
SCHEMBL5504161 0.88 TSHR (0.52) ADORA3ADORA1ADORA2AADORA2BPMP22
SCHEMBL5509065 0.88 TSHR (0.52) ADORA3ADORA1ADORA2AADORA2BPMP22
SCHEMBL5509613 0.88 ADORA3 (0.49) ADORA3ADORA1ADORA2AADORA2BPMP22
SCHEMBL5504164 0.88 TSHR (0.52) ADORA3ADORA1ADORA2AADORA2BPMP22
SCHEMBL5509894 0.88 MEN1 (0.42) PI4KAPI4K2BPI4K2API4KBADORA3
SCHEMBL5509905 0.88 MEN1 (0.42) PI4KAPI4K2BPI4K2API4KBADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537133-B1 PARTIAL AND FULL AGONISTS OF A1 ADENOSINE RECEPTORS CV THERAPEUTICS INC (US) 2007-07-25 EP disclosed