SCHEMBL5504659

SCHEMBL5504659

CC1(C)CN([C@@H](CNC(=O)C(C(N)=O)C2CCCCC2)C2CC2)c2ccc(F)cc21

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.42
SLC6A4 P31645 3/20 0.42
CTSS P25774 14/20 0.40
CTSL P07711 2/20 0.40
CTSK P43235 2/20 0.40
NPC1 O15118 1/20 0.35
POLB P06746 1/20 0.35
RAB9A P51151 1/20 0.35
DPP9 Q86TI2 1/20 0.35
CHRNA7 P36544 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5497674 0.78 CTSS (0.60) CTSSCTSLCTSK
SCHEMBL6687593 0.78 CTSS (0.60) CTSSCTSLCTSK
SCHEMBL4468350 0.72 CTSS (0.71) CTSSCTSLCTSK
SCHEMBL4468345 0.72 CTSS (0.71) CTSSCTSLCTSK
SCHEMBL5408243 0.68 CTSS (0.53) CTSSCTSLCTSKDPP9
SCHEMBL6691416 0.68 CTSS (0.53) CTSSCTSLCTSKDPP9
SCHEMBL6690869 0.67 CTSS (0.60) CTSSCTSLCTSKDPP9
SCHEMBL3023914 0.67 CTSS (0.65) CTSSCTSLCTSK
SCHEMBL27636160 0.66 SLC6A2 (0.49) SLC6A2SLC6A4CTSSCTSLCTSK
SCHEMBL5404869 0.66 CTSS (0.48) CTSSCTSLCTSKNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1658267-A4 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2007-08-01 EP disclosed
EP-1658267-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2006-05-24 EP disclosed
WO-2005034848-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2005-04-21 WO disclosed