SCHEMBL5504840

SCHEMBL5504840

Cn1nnc(-c2ccccc2CC=O)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.41
RAB9A P51151 2/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PDK2 Q15119 1/20 0.41
KDM2B Q8NHM5 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
AGTR1 P30556 1/20 0.35
AGTR2 P50052 1/20 0.35
F2 P00734 1/20 0.34
MAPK8 P45983 1/20 0.33
MAPK10 P53779 1/20 0.33
ATM Q13315 1/20 0.33
EPHX2 P34913 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ABCG2 Q9UNQ0 1/20 0.33
GRM5 P41594 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15238147 0.80 NPC1 (0.44) NPC1RAB9ANFKB1NFKB2RELA
Hydrochloric Acid SCHEMBL5855080 0.78 NPC1 (0.43) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL6189224 0.76 PDK2 (0.44) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL8210469 0.76 IDO1 (0.42) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL13846109 0.72 PDK2 (0.48) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL17198744 0.71 TYK2 (0.45) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL2647877 0.70 PDK2 (0.50) SMN1; SMN2PDK2NPSR1GRM5HPGD
SCHEMBL5855644 0.69 KCNA5 (0.49) NPC1RAB9APDK2F2MAPK8
SCHEMBL7621991 0.69 GABRA1 (0.35)
SCHEMBL5504833 0.69 PDK2 (0.46) NPC1RAB9ASMN1; SMN2PDK2KDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1794157-A1 2-ACYLAMINOTHIAZOLE DERIVATIVES H.Lundbeck A/S (DK) 2007-06-13 EP disclosed
WO-2006032273-A1 2-ACYLAMINOTHIAZOLE DERIVATIVES H. LUNDBECK A/S (DK) 2006-03-30 WO disclosed