SCHEMBL5507510

SCHEMBL5507510

CC(C)(C)n1cc2c(n1)c(=O)n(CO)c1ccccc21

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.48
ALDH1A1 P00352 2/20 0.39
PER2 O15055 5/20 0.38
KDM4E B2RXH2 3/20 0.38
RCE1 Q9Y256 1/20 0.38
PGR P06401 1/20 0.37
RORA P35398 1/20 0.37
RORC P51449 1/20 0.37
RORB Q92753 1/20 0.37
TOP2A P11388 2/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5504756 0.86 ADORA3 (0.47) ADORA3ALDH1A1PER2KDM4ERCE1
SCHEMBL5508801 0.68 ADORA3 (0.83) ADORA3ALDH1A1KDM4ERCE1PGR
SCHEMBL29868746 0.67 CYP1A2 (0.64) ALDH1A1KDM4E
SCHEMBL151036 0.67 CYP1A2 (0.64) ALDH1A1KDM4E
SCHEMBL730877 0.67 ADORA3 (0.58) ADORA3ALDH1A1KDM4ELMNAHPGD
SCHEMBL5511769 0.65 ADORA3 (1.00) ADORA3ALDH1A1KDM4EPGRRORA
SCHEMBL5513775 0.63 ADORA3 (0.86) ADORA3ALDH1A1KDM4EPGRRORA
Hydrochloric Acid SCHEMBL5507703 0.63 ADORA3 (0.71) ADORA3KDM4EPGR
SCHEMBL18539423 0.60 CYP1A2 (0.48) ALDH1A1PER2KDM4E
SCHEMBL11884498 0.60 ERCC1 (0.62) ALDH1A1KDM4EPGRLMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863813-A2 PYRAZOLO[3,4-C]QUINOLINES, PYRAZOLO[3,4-C]NAPHTHYRIDINES, ANALOGS THEREOF, AND METHODS Coley Pharmaceutical Group, Inc. (US) 2007-12-12 EP disclosed
WO-2006107771-A2 PYRAZOLO[3,4-c]QUINOLINES, PYRAZOLO[3,4-c]NAPHTHYRIDINES, ANALOGS THEREOF, AND METHODS COLEY PHARMACEUTICAL GROUP, INC. (US) 2006-10-12 WO disclosed