SCHEMBL5508801

SCHEMBL5508801

CCn1c(=O)c2nn(-c3ccccc3)cc2c2ccccc21

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 10/20 0.83
PGR P06401 2/20 0.52
LMNA P02545 2/20 0.49
HTT P42858 2/20 0.49
HPGD P15428 1/20 0.49
MAPK1 P28482 1/20 0.49
MAPK8 P45983 1/20 0.49
ALDH1A1 P00352 2/20 0.47
CA9 Q16790 1/20 0.47
MAT2A P31153 1/20 0.46
ADORA2A P29274 3/20 0.46
ADORA1 P30542 2/20 0.46
KDM4E B2RXH2 2/20 0.46
RCE1 Q9Y256 1/20 0.46
NPSR1 Q6W5P4 2/20 0.42
NPC1 O15118 1/20 0.42
MITF O75030 1/20 0.42
MAPT P10636 1/20 0.42
AGTR1 P30556 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5511769 0.91 ADORA3 (1.00) ADORA3PGRLMNAHTTHPGD
SCHEMBL5513775 0.89 ADORA3 (0.86) ADORA3PGRLMNAHTTHPGD
Hydrochloric Acid SCHEMBL5507703 0.86 ADORA3 (0.71) ADORA3PGRCA9MAT2AADORA2A
SCHEMBL5509727 0.85 ADORA3 (0.77) ADORA3CA9MAT2AADORA2AADORA1
SCHEMBL5503114 0.83 ADORA3 (1.00) ADORA3PGRHPGDALDH1A1CA9
SCHEMBL5503857 0.77 ADORA3 (0.64) ADORA3HPGDCA9ADORA2AADORA1
SCHEMBL14802110 0.74 ADORA3 (0.55) ADORA3MAPK8CA9ADORA2AADORA1
SCHEMBL11720741 0.73 PGR (0.69) PGRLMNAHTTHPGDMAPK1
SCHEMBL5502979 0.71 HTT (0.51) ADORA3PGRLMNAHTTHPGD
SCHEMBL151563 0.69 ALDH1A1 (0.75) LMNAHTTHPGDMAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863813-A2 PYRAZOLO[3,4-C]QUINOLINES, PYRAZOLO[3,4-C]NAPHTHYRIDINES, ANALOGS THEREOF, AND METHODS Coley Pharmaceutical Group, Inc. (US) 2007-12-12 EP disclosed
WO-2006107771-A2 PYRAZOLO[3,4-c]QUINOLINES, PYRAZOLO[3,4-c]NAPHTHYRIDINES, ANALOGS THEREOF, AND METHODS COLEY PHARMACEUTICAL GROUP, INC. (US) 2006-10-12 WO disclosed