SCHEMBL5513775

SCHEMBL5513775

CCCCn1c(=O)c2nn(-c3ccccc3)cc2c2ccccc21

nearest known ligand 0.86

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.86
PGR P06401 4/20 0.59
RORA P35398 3/20 0.59
RORC P51449 3/20 0.59
RORB Q92753 3/20 0.59
ALDH1A1 P00352 5/20 0.51
PDE4A P27815 1/20 0.48
PDE4B Q07343 1/20 0.48
PDE4C Q08493 1/20 0.48
PDE4D Q08499 1/20 0.48
PDE3B Q13370 1/20 0.48
PDE3A Q14432 1/20 0.48
KDM4E B2RXH2 4/20 0.48
HPGD P15428 3/20 0.48
LMNA P02545 2/20 0.48
CNR2 P34972 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MAPT P10636 1/20 0.46
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5511769 0.93 ADORA3 (1.00) ADORA3PGRRORARORCRORB
SCHEMBL5508801 0.89 ADORA3 (0.83) ADORA3PGRALDH1A1KDM4EHPGD
SCHEMBL5509727 0.85 ADORA3 (0.77) ADORA3KDM4EMAPTSMN1; SMN2
Hydrochloric Acid SCHEMBL5507703 0.81 ADORA3 (0.71) ADORA3PGRKDM4ESMN1; SMN2
SCHEMBL5503114 0.80 ADORA3 (1.00) ADORA3PGRALDH1A1KDM4EHPGD
SCHEMBL5503857 0.77 ADORA3 (0.64) ADORA3KDM4EHPGDCNR2SMN1; SMN2
SCHEMBL14141960 0.75 RORA (1.00) PGRRORARORCRORBALDH1A1
SCHEMBL9209736 0.75 PGR (0.54) ADORA3PGRRORARORCRORB
SCHEMBL9208110 0.72 PGR (0.58) ADORA3PGRRORARORCRORB
SCHEMBL29531665 0.72 PGR (0.73) PGRRORARORCRORBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863813-A2 PYRAZOLO[3,4-C]QUINOLINES, PYRAZOLO[3,4-C]NAPHTHYRIDINES, ANALOGS THEREOF, AND METHODS Coley Pharmaceutical Group, Inc. (US) 2007-12-12 EP disclosed
WO-2006107771-A2 PYRAZOLO[3,4-c]QUINOLINES, PYRAZOLO[3,4-c]NAPHTHYRIDINES, ANALOGS THEREOF, AND METHODS COLEY PHARMACEUTICAL GROUP, INC. (US) 2006-10-12 WO disclosed