SCHEMBL5512657

SCHEMBL5512657

CCC(C(=O)O)c1[nH]nc2c(=O)[nH]c3ccccc3c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.46
KDM4E B2RXH2 8/20 0.39
TDP1 Q9NUW8 1/20 0.39
ALDH1A1 P00352 6/20 0.39
HPGD P15428 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
PARP1 P09874 1/20 0.38
POLB P06746 1/20 0.38
GLA P06280 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 2/20 0.37
HTT P42858 2/20 0.37
ADORA3 P0DMS8 1/20 0.37
NPC1 O15118 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C19 P33261 1/20 0.37
RAB9A P51151 1/20 0.37
MCL1 Q07820 1/20 0.37
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL729439 0.76 ADORA3 (0.40) CHEK1KDM4ETDP1ALDH1A1HPGD
SCHEMBL729000 0.75 ADORA3 (0.41) ALDH1A1HPGDMEN1KMT2APOLB
SCHEMBL731128 0.74 CHEK1 (0.55) CHEK1KDM4EALDH1A1HPGDMEN1
SCHEMBL28250510 0.72 MEN1 (0.43) KDM4EALDH1A1MEN1KMT2APOLB
SCHEMBL29868109 0.70 KDM4E (0.48) KDM4EALDH1A1HPGDPOLBTSHR
SCHEMBL9530036 0.69 POLB (0.67) KDM4EALDH1A1MEN1KMT2APARP1
SCHEMBL9698674 0.66 MEN1 (0.60) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL6601304 0.65 PARP14 (0.46) KDM4EALDH1A1MEN1KMT2AHTT
SCHEMBL28803380 0.65 POLB (0.56) KDM4EALDH1A1KMT2APARP1POLB
SCHEMBL1895662 0.64 ALDH1A1 (0.44) KDM4ETDP1ALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863813-A2 PYRAZOLO[3,4-C]QUINOLINES, PYRAZOLO[3,4-C]NAPHTHYRIDINES, ANALOGS THEREOF, AND METHODS Coley Pharmaceutical Group, Inc. (US) 2007-12-12 EP disclosed
WO-2006107771-A2 PYRAZOLO[3,4-c]QUINOLINES, PYRAZOLO[3,4-c]NAPHTHYRIDINES, ANALOGS THEREOF, AND METHODS COLEY PHARMACEUTICAL GROUP, INC. (US) 2006-10-12 WO disclosed