SCHEMBL5514977

SCHEMBL5514977

CC(C)c1ccc(OCC(=O)O)cc1C(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AGER Q15109 1/20 0.51
PTPN7 P35236 1/20 0.49
THRB P10828 7/20 0.47
THRA P10827 6/20 0.47
MAPT P10636 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
ALDH1A1 P00352 2/20 0.46
TSHR P16473 1/20 0.46
MCL1 Q07820 1/20 0.46
PPARD Q03181 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
LMNA P02545 1/20 0.44
PPARA Q07869 1/20 0.43
SRD5A2 P31213 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21725512 0.82 NQO1 (0.43) MAPTL3MBTL1TSHRLMNA
SCHEMBL5543083 0.81 MCL1 (0.56) AGERPTPN7MAPTL3MBTL1ALDH1A1
SCHEMBL5514421 0.81 PTPN7 (0.53) PTPN7THRBTHRAMAPTL3MBTL1
SCHEMBL17896566 0.79 SMN1; SMN2 (0.55) AGERPTPN7THRBTHRAMAPT
SCHEMBL25063883 0.79 KMT2A (0.48) MAPTALDH1A1SMN1; SMN2LMNA
SCHEMBL585845 0.79 AGER (0.56) AGERPTPN7MAPTL3MBTL1ALDH1A1
SCHEMBL2950207 0.79 MCL1 (0.62) PTPN7THRBTHRAMAPTL3MBTL1
SCHEMBL25725072 0.78 SMN1; SMN2 (0.54) PTPN7THRBTHRAMAPTL3MBTL1
SCHEMBL24935669 0.78 THRA (0.41) THRBTHRAPPARDPPARASRD5A2
SCHEMBL22666573 0.78 THRB (0.61) AGERPTPN7THRBTHRAMCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed