SCHEMBL5515228

SCHEMBL5515228

COC(=O)C(c1cc2ccccc2s1)C(C)C

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 3/20 0.51
CYP1A2 P05177 2/20 0.51
PTGES O14684 1/20 0.51
LMNA P02545 1/20 0.51
LTA4H P09960 1/20 0.51
GAA P10253 1/20 0.51
ALOX15 P16050 1/20 0.51
ALOX12 P18054 1/20 0.51
ALOX5AP P20292 1/20 0.51
LOX P28300 1/20 0.51
EPHX2 P34913 1/20 0.51
PTGS2 P35354 1/20 0.51
LTB4R Q15722 1/20 0.51
TAS1R3 Q7RTX0 2/20 0.50
TAS1R1 Q7RTX1 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14215435 0.85 ALOX5 (0.54) ALOX5CYP1A2PTGESLMNALTA4H
SCHEMBL5511661 0.83 ALOX5 (0.55) ALOX5CYP1A2PTGESLMNALTA4H
SCHEMBL1578437 0.81 ALOX5 (0.49) ALOX5CYP1A2PTGESLMNALTA4H
SCHEMBL2746353 0.81 ALOX5 (0.52) ALOX5CYP1A2PTGESLMNALTA4H
SCHEMBL11491957 0.75 MMP1 (0.43) ALOX5CYP1A2PTGESLMNALTA4H
SCHEMBL11486785 0.75 ALOX5 (0.40) ALOX5CYP1A2PTGESLMNALTA4H
SCHEMBL1666934 0.75 ALOX5 (0.56) ALOX5CYP1A2PTGESLMNALTA4H
SCHEMBL4954902 0.73 TAS1R3 (0.50) ALOX5CYP1A2PTGESLMNALTA4H
SCHEMBL27587691 0.73 TAS1R3 (0.50) ALOX5CYP1A2PTGESLMNALTA4H
SCHEMBL5542170 0.73 ALOX5 (0.57) ALOX5CYP1A2PTGESLMNALTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed