SCHEMBL551705

SCHEMBL551705

C[SiH](C)OCC#CC1=CCCCC1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.36
GRM5 P41594 2/20 0.36
FFAR1 O14842 1/20 0.35
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
CTSK P43235 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
ATM Q13315 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL552152 0.83 CYP1A2 (0.34) CYP1A2GRM5FFAR1ALDH1A1MAPT
SCHEMBL551632 0.71 FFAR1 (0.44) CYP1A2GRM5FFAR1ALDH1A1MAPT
SCHEMBL4212451 0.69
SCHEMBL4222484 0.68
SCHEMBL4098240 0.67 CYP1A2 (0.42) CYP1A2GRM5FFAR1ALDH1A1MAPT
SCHEMBL29080299 0.67 CYP1A2 (0.39) CYP1A2GRM5FFAR1
SCHEMBL28166498 0.67 KCNH2 (0.41) CYP1A2GRM5FFAR1
SCHEMBL7925007 0.64 FFAR1 (0.39) CYP1A2GRM5FFAR1ALDH1A1MAPT
SCHEMBL11744141 0.64
SCHEMBL4854449 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8110695-B2 Compounds and compositions containing silicon and/or other heteroatoms and/or metals and methods of making and using them WELKER MARK E (US) 2012-02-07 US disclosed
US-8110695-B2 Compounds and compositions containing silicon and/or other heteroatoms and/or metals and methods of making and using them WELKER MARK E (US) 2012-02-07 US disclosed
US-20100056801-A1 Compounds And Compositions Containing Silicon And/Or Other Heteroatoms And/Or Metals And Methods of Making And Using Them WELKER MARK E 2010-03-04 US disclosed
US-20100056801-A1 Compounds And Compositions Containing Silicon And/Or Other Heteroatoms And/Or Metals And Methods of Making And Using Them WELKER MARK E 2010-03-04 US disclosed
WO-2008054718-A2 COMPOUNDS AND COMPOSITIONS CONTAINING SILICON AND/OR OTHER HETEROATOMS AND/OR METALS AND METHODS OF MAKING AND USING THEM WAKE FOREST UNIVERSITY (US) 2008-05-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100056801-A1 Compounds And Compositions Containing Silicon And/Or Other Heteroatoms And/Or Metals And Methods of Making And Using Them CA6, SOD1, CA1 CYP1A2 430/4885GRM5 2960/4885FFAR1 4855/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.