SCHEMBL5518997

SCHEMBL5518997

CC(C)(C)OC(=O)NC1=NC(=O)/C(=C/Cc2ccc3nccc(Oc4ccccc4)c3c2)S1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 6/20 0.39
KIT P10721 3/20 0.39
MET P08581 6/20 0.37
KDR P35968 2/20 0.37
BTK Q06187 5/20 0.36
EGFR P00533 4/20 0.36
ERBB2 P04626 1/20 0.34
TEC P42680 1/20 0.34
TXK P42681 1/20 0.34
BLK P51451 1/20 0.34
BMX P51813 1/20 0.34
JAK3 P52333 1/20 0.34
ERBB4 Q15303 1/20 0.34
DDR2 Q16832 1/20 0.34
AXL P30530 1/20 0.34
AAK1 Q2M2I8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5518881 0.90 AAK1 (0.33) PDGFRAKITMETKDRDDR2
SCHEMBL5508606 0.89 PDGFRA (0.39) PDGFRAKITMETKDRBTK
SCHEMBL5509074 0.86 FLT3 (0.33) METAXLAAK1
SCHEMBL5506720 0.86 MET (0.33) METBTKEGFRERBB2TEC
SCHEMBL14437285 0.86 PDGFRA (0.41) PDGFRAKITKDRBTKEGFR
SCHEMBL5506278 0.80 MET (0.36) PDGFRAMETKDRDDR2AXL
SCHEMBL5508442 0.79 MEN1 (0.41) PDGFRAKIT
SCHEMBL5505043 0.78 CLK4 (0.36) AXL
SCHEMBL5510840 0.77 MET (0.36) METBTKEGFRERBB2TEC
SCHEMBL14437267 0.75 CISD1 (0.40) AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7253285-B2 Thiazolinone 4-monosubstituted quinolines HOFFMANN-LA ROCHE INC. (US) 2007-08-07 US disclosed
US-20060063805-A1 Thiazolinone 4-monosubstituted quinolines CHEN LI 2006-03-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060063805-A1 Thiazolinone 4-monosubstituted quinolines CDK1, CDK14, CDK17 PDGFRA 3386/4885KIT 2841/4885MET 1954/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.