SCHEMBL5520722

SCHEMBL5520722

C=C[C](c1ccccc1)c1cccc2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A1 P22736 1/20 0.50
NR4A2 P43354 1/20 0.50
NR4A3 Q92570 1/20 0.50
CDC25B P30305 1/20 0.44
PTK2B Q14289 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MMP3 P08254 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
ALDH1A1 P00352 2/20 0.41
PTPN1 P18031 1/20 0.41
PLK1 P53350 1/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
AKT1 P31749 1/20 0.39
CYP1A2 P05177 3/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
GPR52 Q9Y2T5 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14977560 0.88 NR4A1 (0.52) NR4A1NR4A2NR4A3CDC25BPTK2B
SCHEMBL84200 0.75 AKT1 (0.56) L3MBTL1ALDH1A1HPGDSMN1; SMN2AKT1
SCHEMBL9422531 0.75 AKT1 (0.56) L3MBTL1ALDH1A1HPGDSMN1; SMN2AKT1
SCHEMBL31371895 0.75 NR4A1 (0.55) NR4A1NR4A2NR4A3CDC25BPTK2B
SCHEMBL7941531 0.75 PTK2B (0.52) NR4A1NR4A2NR4A3CDC25BPTK2B
SCHEMBL1933651 0.75 NR4A1 (0.55) NR4A1NR4A2NR4A3CDC25BPTK2B
SCHEMBL5012386 0.74 NR4A1 (0.59) NR4A1NR4A2NR4A3CDC25BPTK2B
SCHEMBL40515 0.74 NR4A1 (0.59) NR4A1NR4A2NR4A3CDC25BPTK2B
SCHEMBL29465774 0.73 NR4A1 (0.59) NR4A1NR4A2NR4A3CDC25BPTK2B
SCHEMBL726189 0.73 NR4A1 (0.59) NR4A1NR4A2NR4A3CDC25BPTK2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1754475-A1 Use of C-terminal modified oxamyl dipeptides as inhibitors of the ice/ced-3 family of cysteine proteases Idun Pharmaceuticals, Inc. (US) 2007-02-21 EP claimed
JP-3815968-B2 2006-08-30 JP claimed
JP-2002519406-A 2002-07-02 JP claimed
EP-1091930-A1 C-TERMINAL MODIFIED OXAMYL DIPEPTIDES AS INHIBITORS OF THE ICE/ced-3 FAMILY OF CYSTEINE PROTEASES Idun Pharmaceuticals, Inc. (US) 2001-04-18 EP claimed
WO-2000001666-A1 C-TERMINAL MODIFIED OXAMYL DIPEPTIDES AS INHIBITORS OF THE ICE/ced-3 FAMILY OF CYSTEINE PROTEASES IDUN PHARMACEUTICALS, INC. (US) 2000-01-13 WO claimed