SCHEMBL5524975

SCHEMBL5524975

CC(C)(C)OC(=O)OC(=O)CC1CNC(c2ccc(C(N)=NO)cc2)C1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
MAPK1 P28482 1/20 0.38
POLB P06746 1/20 0.35
S1PR4 O95977 8/20 0.34
S1PR1 P21453 8/20 0.34
S1PR5 Q9H228 8/20 0.34
S1PR3 Q99500 5/20 0.34
MASP2 O00187 2/20 0.33
GAA P10253 1/20 0.30
RAB9A P51151 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5530479 0.82 GPR119 (0.36) S1PR4S1PR1S1PR5S1PR3
SCHEMBL5524979 0.73 MASP2 (0.36) KMT2AMEN1MAPK1MASP2
SCHEMBL3496764 0.69 MEN1 (0.37) KMT2AMEN1MAPK1POLB
SCHEMBL3496771 0.69 MEN1 (0.37) KMT2AMEN1MAPK1POLB
SCHEMBL3496769 0.69 MEN1 (0.37) KMT2AMEN1MAPK1POLB
SCHEMBL3496766 0.69 MEN1 (0.37) KMT2AMEN1MAPK1POLB
SCHEMBL3497056 0.69 MEN1 (0.37) KMT2AMEN1MAPK1POLB
SCHEMBL3497055 0.69 MEN1 (0.37) KMT2AMEN1MAPK1POLB
SCHEMBL3497054 0.69 MEN1 (0.37) KMT2AMEN1MAPK1POLB
SCHEMBL3497061 0.69 MEN1 (0.37) KMT2AMEN1MAPK1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1804793-A2 2-(ARYL)AZACYCLYLMETHYL CARBOXYLATES, SULFONATES, PHOSPHONATES, PHOSPHINATES AND HETEROCYCLES AS S1P RECEPTOR AGONISTS Merck & Co., Inc. (US) 2007-07-11 EP disclosed
WO-2006047195-A2 2-(ARYL)AZACYCLYLMETHYL CARBOXYLATES, SULFONATES, PHOSPHONATES, PHOSPHINATES AND HETEROCYCLES AS S1P RECEPTOR AGONISTS MERCK & CO., INC. (US) 2006-05-04 WO disclosed