SCHEMBL5524979

SCHEMBL5524979

CC(C)(C)OC(=O)C(C(=O)O)C1CNC(c2ccc(C(N)=NO)cc2)C1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MASP2 O00187 2/20 0.36
MEN1 O00255 1/20 0.34
MAPK1 P28482 1/20 0.34
KMT2A Q03164 1/20 0.34
ITGB3 P05106 1/20 0.31
ITGA2B P08514 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5530482 0.82 GPR119 (0.34)
SCHEMBL5524975 0.73 KMT2A (0.38) MASP2MEN1MAPK1KMT2A
SCHEMBL5135071 0.66 KMT2A (0.34) MEN1MAPK1KMT2A
SCHEMBL5527997 0.65 PTGES (0.37) MEN1KMT2AITGB3ITGA2B
SCHEMBL31581462 0.64 CTSS (0.47) MEN1KMT2AITGB3ITGA2B
SCHEMBL27192552 0.63 CHRM2 (0.33) MEN1KMT2A
SCHEMBL21001140 0.62 GPR119 (0.42) MEN1MAPK1KMT2AITGB3ITGA2B
SCHEMBL12385571 0.61 GRIN2B (0.34) MEN1MAPK1KMT2AITGB3ITGA2B
SCHEMBL2296923 0.61 GRIN2B (0.34) MEN1MAPK1KMT2AITGB3ITGA2B
SCHEMBL29120582 0.61 CPN1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1804793-A2 2-(ARYL)AZACYCLYLMETHYL CARBOXYLATES, SULFONATES, PHOSPHONATES, PHOSPHINATES AND HETEROCYCLES AS S1P RECEPTOR AGONISTS Merck & Co., Inc. (US) 2007-07-11 EP disclosed
WO-2006047195-A2 2-(ARYL)AZACYCLYLMETHYL CARBOXYLATES, SULFONATES, PHOSPHONATES, PHOSPHINATES AND HETEROCYCLES AS S1P RECEPTOR AGONISTS MERCK & CO., INC. (US) 2006-05-04 WO disclosed